SCHEMBL3665283

SCHEMBL3665283

CC(C)(N)CSCC(=O)c1ccc2[nH]c3nc(Cl)ccc3c2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.35
CA1 P00915 7/20 0.34
CA2 P00918 7/20 0.34
CA7 P43166 7/20 0.34
CA13 Q8N1Q1 7/20 0.34
CA12 O43570 6/20 0.34
CA6 P23280 6/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.33
POLB P06746 1/20 0.33
CA9 Q16790 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL675929 0.83 MAP2 (0.36) KIF11CA1CA2CA7CA13
Diethylamine SCHEMBL3664811 0.82 HDAC3 (0.35) KIF11CA1CA2CA7CA13
SCHEMBL3665277 0.82 MAPT (0.33) KIF11NPC1RAB9AHDAC3HDAC1
SCHEMBL3665281 0.81 KDM4E (0.39) HDAC3HDAC1HDAC2HDAC6HDAC5
SCHEMBL675224 0.81 ALDH1A1 (0.38) CA1CA2CA7CA13NPC1
SCHEMBL3668534 0.80 ERBB2 (0.42) CA1CA2CA7CA13CA12
SCHEMBL678686 0.80 TERT (0.35) RAB9AHDAC3HDAC1HDAC2HDAC6
SCHEMBL3665280 0.79 KIF11 (0.34) KIF11NPC1RAB9AHDAC3HDAC1
SCHEMBL675108 0.78 CA1 (0.46) CA1CA2CA7CA13NPC1
SCHEMBL676048 0.77 GSK3B (0.41) KIF11RAB9ACYP1A2CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed