SCHEMBL367120

SCHEMBL367120

CS(=O)(=O)NC(=O)c1ccc(OCc2ccc(Cl)cc2)c(C#N)c1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
XDH P47989 3/20 0.54
SCN9A Q15858 5/20 0.53
SCN5A Q14524 3/20 0.53
SMPD1 P17405 1/20 0.52
MRGPRX4 Q96LA9 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366522 0.89 MRGPRX4 (0.56) HDAC1SCN9ASCN5AMRGPRX4
SCHEMBL364527 0.85 SCN9A (0.63) HDAC8HDAC1HDAC6SCN9ASCN5A
SCHEMBL364759 0.81 MRGPRX4 (0.64) HDAC8HDAC1HDAC6SCN9ASCN5A
SCHEMBL16240302 0.79 MRGPRX4 (0.61) HDAC8HDAC1HDAC6SCN9ASCN5A
SCHEMBL16319800 0.78 SCN9A (0.59) SCN9ASCN5A
SCHEMBL365210 0.78 MAOA (0.63) SCN9ASCN5A
SCHEMBL366081 0.78 MAOA (0.63) SCN9ASCN5A
SCHEMBL365866 0.77 SCN9A (0.49) XDHSCN9ASCN5A
SCHEMBL369367 0.77 CYP19A1 (0.45) SCN9ASCN5AMRGPRX4
Diethylamine SCHEMBL16239865 0.76 MRGPRX4 (0.58) HDAC8HDAC1HDAC6SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A HDAC8 925/4885HDAC1 370/4885HDAC6 556/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.