SCHEMBL367237

SCHEMBL367237

COc1cc(OC(=O)N2CCOCC2)cn2c1c(C(N)=O)c1ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
RAB9A P51151 3/20 0.45
NPC1 O15118 2/20 0.45
TP53 P04637 1/20 0.44
GAA P10253 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
EPHX1 P07099 2/20 0.43
HSD17B10 Q99714 1/20 0.43
KMT2A Q03164 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
GLA P06280 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 2/20 0.41
USP2 O75604 1/20 0.41
CASP3 P42574 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366114 0.91 TSHR (0.47) TSHRL3MBTL1RAB9ANPC1TP53
SCHEMBL365264 0.87 EPHX1 (0.45) TSHRL3MBTL1RAB9ANPC1TP53
SCHEMBL365101 0.81 KMT2A (0.51) TSHRRAB9ANPC1TP53GAA
SCHEMBL365490 0.80 NCEH1 (0.39) TSHRRAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL367409 0.78 EPHX1 (0.48) TSHRRAB9ANPC1TP53GAA
SCHEMBL367236 0.78 TSHR (0.47) TSHRL3MBTL1RAB9ANPC1TP53
SCHEMBL366075 0.77 MAPT (0.35) L3MBTL1TP53NPSR1KMT2ASMN1; SMN2
SCHEMBL365192 0.76 EGFR (0.41) TSHRL3MBTL1GAANPSR1KMT2A
SCHEMBL367766 0.76 L3MBTL1 (0.43) TSHRL3MBTL1RAB9ANPC1NPSR1
SCHEMBL367225 0.75 KMT2A (0.40) TSHRNPC1NPSR1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed