SCHEMBL367409

SCHEMBL367409

O=C(O)c1c2ccccc2n2cc(OC(=O)N3CCOCC3)cc(O)c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.48
HSD17B10 Q99714 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
KMT2A Q03164 3/20 0.48
NPC1 O15118 2/20 0.48
KDM4E B2RXH2 1/20 0.48
RAB9A P51151 1/20 0.48
MEN1 O00255 1/20 0.46
CASP3 P42574 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAOB P27338 1/20 0.42
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365264 0.91 EPHX1 (0.45) EPHX1HSD17B10SMN1; SMN2KMT2ANPC1
SCHEMBL366114 0.87 TSHR (0.47) EPHX1HSD17B10SMN1; SMN2KMT2ANPC1
SCHEMBL365668 0.83 KMT2A (0.55) EPHX1HSD17B10SMN1; SMN2KMT2ANPC1
SCHEMBL367237 0.78 TSHR (0.49) EPHX1HSD17B10SMN1; SMN2KMT2ANPC1
SCHEMBL365213 0.77 PKM (0.39) KMT2ANPC1RAB9AMEN1TSHR
SCHEMBL366116 0.75 CA1 (0.41)
SCHEMBL365101 0.75 KMT2A (0.51) EPHX1HSD17B10SMN1; SMN2KMT2ANPC1
SCHEMBL367408 0.75 EPHX1 (0.51) EPHX1HSD17B10SMN1; SMN2KMT2ANPC1
SCHEMBL365667 0.74 EPHX1 (0.56) EPHX1HSD17B10SMN1; SMN2KMT2ANPC1
SCHEMBL367390 0.74 AGTR1 (0.34) SMN1; SMN2KMT2AKDM4EMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed