SCHEMBL3675346

SCHEMBL3675346

CCOC(=O)c1cc2cc(OS(=O)(=O)C(F)(F)F)ccc2n1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 6/20 0.43
NOD1 Q9Y239 6/20 0.43
MAOA P21397 1/20 0.40
ADORA1 P30542 1/20 0.39
LGALS8 O00214 1/20 0.38
LGALS3 P17931 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ELANE P08246 1/20 0.38
HSD11B1 P28845 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
STS P08842 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PPARG P37231 1/20 0.36
PTGS2 P35354 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2813774 0.88 NOD2 (0.40) NOD2NOD1MAOAADORA1LGALS8
SCHEMBL3675353 0.85 KDM4E (0.42) ADORA1LGALS8LGALS3MEN1KMT2A
SCHEMBL3673992 0.80 HSD11B1 (0.42) HSD11B1ALDH1A1HPGDL3MBTL1KDM4E
SCHEMBL3637425 0.78 NOD2 (0.50) NOD2NOD1MAOAMEN1KMT2A
SCHEMBL3639123 0.77 SRD5A2 (0.61) NOD2NOD1MAOAMEN1KMT2A
SCHEMBL5865527 0.77 STS (0.52) HSD11B1ALDH1A1HPGDSTSKDM4E
SCHEMBL3634756 0.76 MAOA (0.45) NOD2NOD1MAOAMEN1KMT2A
SCHEMBL7470558 0.75 NOD2 (0.40) NOD2NOD1MAOALGALS8LGALS3
SCHEMBL8613925 0.74 TSHR (0.47) ADORA1KMT2AHSD11B1ALDH1A1HPGD
SCHEMBL3638008 0.73 NOD2 (0.53) NOD2NOD1ELANEALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170072-A1 FARNESOID X RECEPTOR AGONISTS GlaxoSmithKline LLC (US) 2010-04-07 EP disclosed
WO-2008157270-A1 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed