SCHEMBL368251

SCHEMBL368251

Cc1c(Cl)cccc1S(=O)(=O)Nc1nc(CC(=O)N2CCN(C)CC2)cs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 1.00
HSD17B1 P14061 2/20 1.00
HSD17B2 P37059 2/20 1.00
F2 P00734 3/20 0.47
F10 P00742 3/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
LMNA P02545 1/20 0.44
ALDH1A1 P00352 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALK Q9UM73 1/20 0.42
CTPS1 P17812 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30044126 0.99 HSD11B1 (1.00) HSD11B1HSD17B1HSD17B2F2F10
Hydrochloric Acid SCHEMBL5692696 0.99 HSD11B1 (1.00) HSD11B1HSD17B1HSD17B2F2F10
Trifluoroacetic Acid SCHEMBL3619340 0.94 HSD11B1 (0.89) HSD11B1HSD17B1HSD17B2F2F10
SCHEMBL3616863 0.93 HSD11B1 (0.86) HSD11B1HSD17B1HSD17B2F2F10
SCHEMBL3606652 0.93 HSD11B1 (0.86) HSD11B1HSD17B1HSD17B2F2F10
SCHEMBL16325423 0.92 HSD11B1 (0.85) HSD11B1HSD17B1HSD17B2F2F10
SCHEMBL3616943 0.92 HSD11B1 (0.84) HSD11B1HSD17B1HSD17B2F2F10
SCHEMBL3614188 0.91 HSD11B1 (0.83) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL5692940 0.90 HSD11B1 (0.82) HSD11B1HSD17B1HSD17B2F2F10
SCHEMBL3615493 0.90 HSD11B1 (0.82) HSD11B1HSD17B1HSD17B2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 435 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050137209-A1 Treatment of neurologic disorders with inhibitors of 11beta-HSD1 AGY THERAPEUTICS, INC. 2005-06-23 US claimed
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US disclosed
US-20260137660-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US disclosed
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US disclosed
US-20260137658-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US disclosed
US-20260137659-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US disclosed
US-20250319072-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2025-10-16 US disclosed
EP-4381284-B1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH ZUERICH (CH) 2025-07-09 EP disclosed
US-12329745-B2 Methods and compositions for treating glucocorticoid excess SPARROW PHARMACEUTICALS, INC. (US) 2025-06-17 US disclosed
US-20240293375-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS FIRST-CITIZENS BANK & TRUST COMPANY 2024-09-05 US disclosed
WO-2007039177-A2 PHENYL- AND PYRIDINYL- 1, 2 , 4 - OXADIAZOLONE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
WO-2007039175-A1 N-[1 ,3,4]-THIADIAZOL-2-YL-BENZENE SULFONAMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
WO-2007039171-A1 4-OXY-N-[1 ,3,4]-THIADIAZOL-2-YL-BENZENE SULFONAMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
WO-2007039174-A2 BICYCLIC ARYL-SULFONIC ACID [1,3,4]-THIADIAZOL-2-YL-AMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
WO-2007039176-A1 DERIVATIVES OF 2 -AMINTHIAZOLES AND 2-AMINOOXAZOLES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
WO-2007039178-A2 PHENYL-[1,2,4]-OXADIAZOL-5-ONE DERIVATIVES WITH PHENYL GROUP, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
WO-2007039172-A1 PHENYL- AND PYRIDYL-I, 2 , 4 -OXADIAZOLONE DERIVATIVES WITH PHENYL GROUP, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
WO-2007039173-A1 CYCLIC N-[1 ,3,4]-THIADIAZOL-2-YL-BENZENE SULFONAMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed
US-20050186659-A1 Methods for protein purification BIOVITRUM AB (SE) 2005-08-25 US disclosed
US-20050137209-A1 Treatment of neurologic disorders with inhibitors of 11beta-HSD1 AGY THERAPEUTICS, INC. 2005-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240293375-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS HSD11B1, HSD17B1, HSD3B1 HSD11B1 1/4885HSD17B1 2/4885HSD17B2 4/4885
US-20050137209-A1 Treatment of neurologic disorders with inhibitors of 11beta-HSD1 HSD11B1, HSD17B1, HSD3B1 HSD11B1 1/4885HSD17B1 2/4885HSD17B2 7/4885
US-20250319072-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS HSD11B1, HSD17B1, HSD3B1 HSD11B1 1/4885HSD17B1 2/4885HSD17B2 4/4885
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS NR3C1, NR3C2, SHBG HSD11B1 4/4885HSD17B1 7/4885HSD17B2 13/4885
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS NR3C2, NR3C1, MC2R HSD11B1 4/4885HSD17B1 10/4885HSD17B2 12/4885
US-12329745-B2 Methods and compositions for treating glucocorticoid excess HSD11B1, HSD17B1, HSD3B1 HSD11B1 1/4885HSD17B1 2/4885HSD17B2 4/4885
US-20260137660-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS NR3C1, NR3C2, SHBG HSD11B1 4/4885HSD17B1 9/4885HSD17B2 11/4885
US-20260137659-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS NR3C2, NR3C1, MC2R HSD11B1 4/4885HSD17B1 13/4885HSD17B2 20/4885
US-20260137658-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS NR3C1, NR3C2, NR5A1 HSD11B1 5/4885HSD17B1 7/4885HSD17B2 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.