SCHEMBL3701029

SCHEMBL3701029

CCOC(=O)CN(CCc1c[nH]c2ccccc12)C(=O)CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1CCCN1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 5/20 0.45
MC4R P32245 2/20 0.37
MC5R P33032 2/20 0.37
MC3R P41968 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
APAF1 O14727 3/20 0.36
CASP3 P42574 3/20 0.36
CASP9 P55211 3/20 0.36
CYCS P99999 3/20 0.36
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ACHE P22303 1/20 0.35
TACR1 P25103 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3697589 0.92 BCHE (0.37) TACR2ACHEKDM4E
SCHEMBL3700997 0.89 APAF1 (0.38) MC4RMC5RMC3RAPAF1CASP3
SCHEMBL3705051 0.89 APAF1 (0.36) TACR2APAF1CASP3CASP9CYCS
SCHEMBL3693162 0.87 MAPT (0.37) APAF1CASP3CASP9CYCSDRD2
SCHEMBL3697424 0.87 APAF1 (0.34) TACR2APAF1CASP3CASP9CYCS
SCHEMBL9105301 0.87 TACR2 (0.42) TACR2MC4RMC5RMC3RHRH3
SCHEMBL3705169 0.86 ALDH1A1 (0.36) TACR2APAF1CASP3CASP9CYCS
SCHEMBL9101546 0.85 C5AR1 (0.39) TACR2APAF1CASP3CASP9CYCS
SCHEMBL3696385 0.85 PTGS2 (0.37) HRH3APAF1CASP3CASP9CYCS
SCHEMBL3701027 0.84 APAF1 (0.53) TACR2MC4RMC5RMC3RAPAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9040701-B2 Apaf-1 inhibitor compounds LABORATORIOS SALVAT, S.A. (ES) 2015-05-26 US disclosed
US-20120122868-A1 APAF-1 INHIBITOR COMPOUNDS LABORATORIOS SALVAT, S.A. (ES) 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122868-A1 APAF-1 INHIBITOR COMPOUNDS APAF1, API5, AIFM1 TACR2 4560/4885MC4R 4827/4885MC5R 4593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.