SCHEMBL370059

SCHEMBL370059

Cc1cc(Cl)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(Oc2ccc(Cl)c(C(=O)O)c2)cc1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.35
ADRB3 P13945 3/20 0.34
ADRB1 P08588 2/20 0.34
FFAR1 O14842 2/20 0.33
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
FNTA P49354 1/20 0.31
FNTB P49356 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
BRD4 O60885 1/20 0.31
CHEK2 O96017 1/20 0.30
P2RX3 P56373 1/20 0.30
PRKAB2 O43741 1/20 0.30
PRKAG1 P54619 1/20 0.30
PRKAA2 P54646 1/20 0.30
PRKAA1 Q13131 1/20 0.30
PRKAG3 Q9UGI9 1/20 0.30
PRKAG2 Q9UGJ0 1/20 0.30
PRKAB1 Q9Y478 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363628 0.93 ADRB1 (0.35) GPBAR1ADRB3ADRB1FFAR1FNTA
SCHEMBL363129 0.90 FFAR1 (0.34) GPBAR1ADRB3ADRB1FFAR1CHEK2
SCHEMBL365756 0.89 ADRB3 (0.38) GPBAR1ADRB3ADRB1P2RX3
SCHEMBL365274 0.85 GPBAR1 (0.46) GPBAR1TDP1BRD4
SCHEMBL1389755 0.83 GPBAR1 (0.36) GPBAR1ADRB3ADRB1FFAR1ALDH1A1
SCHEMBL1389758 0.83 GPBAR1 (0.36) GPBAR1ADRB3ADRB1FFAR1ALDH1A1
SCHEMBL363178 0.83 GPBAR1 (0.51) GPBAR1ADRB3ADRB1TDP1BRD4
SCHEMBL362064 0.82 CNR1 (0.37) GPBAR1FFAR1TDP1
SCHEMBL12505651 0.80 GPBAR1 (0.35) GPBAR1BRD4
SCHEMBL365294 0.79 GPBAR1 (0.35) GPBAR1ALDH1A1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed