Dobesilic Acid

Dobesilic Acid

SCHEMBL370202

O=S(=O)(O)c1cc(O)ccc1O.[KH].[KH]

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.70
HSD17B10 Q99714 3/20 0.70
HPGD P15428 1/20 0.70
HIF1A Q16665 1/20 0.70
PTGS1 P23219 1/20 0.61
EGFR P00533 1/20 0.56
GAA P10253 3/20 0.55
POLB P06746 2/20 0.55
GFER P55789 1/20 0.55
ALPL P05186 1/20 0.53
ALPI P09923 1/20 0.53
ALPG P10696 1/20 0.53
DNMT1 P26358 1/20 0.53
MCL1 Q07820 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
ALDH1A1 P00352 3/20 0.49
PKM P14618 1/20 0.49
MPL P40238 2/20 0.43
NSD2 O96028 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dobesilic Acid SCHEMBL78222 1.00 LMNA (0.70) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL232087 0.98 LMNA (0.72) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL29389625 0.98 LMNA (0.72) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL9790423 0.95 LMNA (0.70) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL10589964 0.95 HSD17B10 (0.70) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL344443 0.95 LMNA (0.70) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL214799 0.95 LMNA (0.70) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL78224 0.95 LMNA (0.70) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL15364076 0.95 LMNA (0.70) LMNAHSD17B10HPGDHIF1APTGS1
Dobesilic Acid SCHEMBL866670 0.95 LMNA (0.70) LMNAHSD17B10HPGDHIF1APTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110257264-A1 USE OF 2,5-DIHYDROXYBENZENE DERIVATIVES FOR TREATING ACTINIC KERATOSIS ACTION MEDICINES (ES) 2011-10-20 US claimed
US-20110196040-A1 Skin Penetration Enhancing Systems for Polar Drugs ACTION MEDICINES S.L. (ES) 2011-08-11 US claimed
US-20120077785-A1 METHODS OF USE FOR 2,5-DIHYDROXYBENZENE SULFONIC ACID COMPOUNDS FOR THE TREATMENT OF CANCER, ROSACEA AND PSORIASIS ACTION MEDICINES (ES) 2012-03-29 US disclosed
US-20120015912-A1 USE OF 2,5-DIHYDROXYBENZENE FOR THE TREATMENT OF OCULAR DISEASES ACTION MEDICINES (ES) 2012-01-19 US disclosed
US-20110257264-A1 USE OF 2,5-DIHYDROXYBENZENE DERIVATIVES FOR TREATING ACTINIC KERATOSIS ACTION MEDICINES (ES) 2011-10-20 US disclosed
US-20110196040-A1 Skin Penetration Enhancing Systems for Polar Drugs ACTION MEDICINES S.L. (ES) 2011-08-11 US disclosed
US-20110152222-A1 USE OF 2,5-DIHYDROXYBENZENE DERIVATIVES FOR THE TREATMENT OF ARTHRITIS AND PAIN SANCHEZ PEDRO CUEVAS 2011-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120077785-A1 METHODS OF USE FOR 2,5-DIHYDROXYBENZENE SULFONIC ACID COMPOUNDS FOR THE TREATMENT OF CANCER, ROSACEA AND PSORIASIS IL2, IL2RA, IL5 LMNA 4181/4885HSD17B10 1497/4885HPGD 2149/4885
US-20110196040-A1 Skin Penetration Enhancing Systems for Polar Drugs ABCB11, KCNK5, KCNQ5 LMNA 3019/4885HSD17B10 2486/4885HPGD 2531/4885
US-20120015912-A1 USE OF 2,5-DIHYDROXYBENZENE FOR THE TREATMENT OF OCULAR DISEASES ALDH1A2, CRYAB, HSD17B14 LMNA 2802/4885HSD17B10 104/4885HPGD 134/4885
US-20110257264-A1 USE OF 2,5-DIHYDROXYBENZENE DERIVATIVES FOR TREATING ACTINIC KERATOSIS CYP8B1, DERA, KRT18 LMNA 1346/4885HSD17B10 125/4885HPGD 212/4885
US-20110152222-A1 USE OF 2,5-DIHYDROXYBENZENE DERIVATIVES FOR THE TREATMENT OF ARTHRITIS AND PAIN CYP8B1, CYP26B1, UGT2B7 LMNA 3452/4885HSD17B10 117/4885HPGD 137/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.