SCHEMBL370726

SCHEMBL370726

CCCc1c(C(N)=O)cccc1-c1ccccc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.45
CXCR5 P32302 2/20 0.41
BCAT2 O15382 1/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
LMNA P02545 2/20 0.39
CYP3A4 P08684 2/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
NR1I2 O75469 1/20 0.39
CHRM2 P08172 1/20 0.39
ADRA2A P08913 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065283 0.88 MYC (0.47) MYCBCAT2KEAP1NFE2L2LMNA
SCHEMBL370920 0.86 MYC (0.54) MYCCXCR5LMNACYP3A4MEN1
SCHEMBL4235369 0.85 CXCR5 (0.49) MYCCXCR5LMNACYP3A4MAPT
SCHEMBL5478290 0.84 PARP1 (0.45) BCAT2KEAP1NFE2L2LMNACYP3A4
SCHEMBL5476512 0.83 BCAT2 (0.59) BCAT2KEAP1NFE2L2LMNACYP3A4
SCHEMBL5478916 0.82 MEN1 (0.44) BCAT2KEAP1NFE2L2MEN1KMT2A
SCHEMBL2964481 0.82 PARP1 (0.45) BCAT2KEAP1NFE2L2LMNACYP3A4
SCHEMBL5482149 0.81 MYC (0.47) MYCBCAT2KEAP1NFE2L2MAPT
SCHEMBL5482646 0.81 PPARG (0.45) BCAT2MAPTALDH1A1HPGDPPARG
SCHEMBL5742619 0.80 MYC (0.53) MYCBCAT2KEAP1NFE2L2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed