SCHEMBL3710928

SCHEMBL3710928

C=CCN1C(=O)C2CCC1(N(Cc1ccc(S(=O)(=O)CCC)cc1)C(=O)O)CC2

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.33
TAS2R14 Q9NYV8 1/20 0.30
ALDH1A1 P00352 1/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4186270 0.83 NPC1 (0.36) ALDH1A1OPRD1
SCHEMBL3786553 0.82 RORC (0.32) RORCALDH1A1OPRD1
SCHEMBL3710931 0.79 OPRM1 (0.31) OPRD1
SCHEMBL3709702 0.75 SLC6A9 (0.41) RORC
SCHEMBL4243962 0.65 OPRD1 (0.34) OPRD1
SCHEMBL3786554 0.65 OPRM1 (0.32) ALDH1A1OPRD1
SCHEMBL4181995 0.63 NPC1 (0.36) OPRD1
SCHEMBL3711027 0.62 SLC6A9 (0.44) RORC
SCHEMBL3704054 0.61 SLC6A9 (0.47)
SCHEMBL4243958 0.60 OXTR (0.34) OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010087761-A1 2-AZA-BICYCLO[2.2.2]OCTANE COMPOUNDS AND USES THEREOF ASTRAZENECA AB (SE) 2010-08-05 WO disclosed