SCHEMBL3711048

SCHEMBL3711048

CCOC(=O)N(c1ccccc1Cl)c1c(C)noc1-c1ccc(-c2cccc(C(=O)O)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
P2RY12 Q9H244 2/20 0.35
CTSA P10619 3/20 0.35
MAPT P10636 4/20 0.34
CNR2 P34972 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
ACR P10323 1/20 0.33
LPAR1 Q92633 1/20 0.33
LPAR2 Q9HBW0 1/20 0.33
LPAR3 Q9UBY5 1/20 0.33
SLC26A6 Q9BXS9 1/20 0.33
DHODH Q02127 1/20 0.32
BRS3 P32247 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3707635 0.93 CTSA (0.35) ALDH1A1KDM4EHPGDSMN1; SMN2P2RY12
SCHEMBL3704916 0.93 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDSMN1; SMN2P2RY12
SCHEMBL1246290 0.87 SCN9A (0.40) ALDH1A1KDM4EHPGDP2RY12CTSA
SCHEMBL3710286 0.86 MAPT (0.40) ALDH1A1KDM4EHPGDSMN1; SMN2MAPT
SCHEMBL2335317 0.85 LPAR1 (0.38) ALDH1A1KDM4EHPGDSMN1; SMN2LPAR1
SCHEMBL3700514 0.85 LPAR1 (0.37) ALDH1A1KDM4EHPGDSMN1; SMN2CTSA
SCHEMBL2336114 0.85 LTB4R2 (0.37) ALDH1A1KDM4EHPGDSMN1; SMN2ACR
SCHEMBL3708659 0.84 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2MAPTLPAR1
SCHEMBL3711161 0.83 LDHA (0.41) ALDH1A1KDM4EHPGDSMN1; SMN2MAPT
SCHEMBL2336147 0.83 NR1H4 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010077882-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-07-08 WO claimed
WO-2010077882-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-07-08 WO disclosed