SCHEMBL3712685

SCHEMBL3712685

CC(C)n1nnc(CCNC(=O)O)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 2/20 0.34
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
GRIK1 P39086 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
CLK1 P49759 1/20 0.32
CLK2 P49760 1/20 0.32
PI4KB Q9UBF8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1778197 0.69 HSD17B10 (0.61) MEN1KMT2AKDM4E
SCHEMBL3712362 0.69 CYP1A2 (0.46) DAGLACYP2D6CYP2C19MEN1CYP1A2
SCHEMBL18839792 0.69 USP2 (0.40) MEN1KMT2AKDM4E
SCHEMBL18839781 0.68 PKM (0.34)
SCHEMBL12662755 0.67 PIK3CD (0.41) PIK3CDPIK3CAPIK3CBPIK3CGCLK1
SCHEMBL5618142 0.66 TSHR (0.40) DAGLATRPV1KDM4E
SCHEMBL14417042 0.65 GRIK1 (0.36) MEN1KMT2AGRIK1GRIA1GRIA2
SCHEMBL5996863 0.65 ALDH1A1 (0.36) DAGLAKMT2AGRIK1GRIA1GRIA2
SCHEMBL22455534 0.65 RAB9A (0.48) CYP2D6
SCHEMBL19347393 0.65 KMT2A (0.39) KMT2APIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed