SCHEMBL3714028

SCHEMBL3714028

Cc1c(-c2ccccc2)ccc(NCc2ccccc2)c1C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 2/20 0.46
CD38 P28907 1/20 0.44
RPS6KB1 P23443 2/20 0.44
CDC7 O00311 1/20 0.44
ROCK2 O75116 1/20 0.44
MAP4K4 O95819 1/20 0.44
GSK3B P49841 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
AKT1 P31749 1/20 0.43
IDO1 P14902 1/20 0.42
PLA2G1B P04054 1/20 0.42
AR P10275 1/20 0.42
HDAC8 Q9BY41 2/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
JAK2 O60674 2/20 0.41
JAK1 P23458 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3698514 0.86 FABP4 (0.40) ALDH1A1HPGDKDM4EMKNK2IDO1
SCHEMBL3704897 0.84 IDO1 (0.42) ALDH1A1HPGDKDM4EIDO1PLA2G1B
SCHEMBL3708760 0.82 KDM4E (0.47) ALDH1A1HPGDKDM4ERPS6KB1HDAC8
SCHEMBL3135452 0.75 BCAT2 (0.47) ALDH1A1HPGDKDM4EBCAT2HSD17B10
SCHEMBL3714031 0.74 AR (0.48) ALDH1A1HPGDKDM4ECD38CDC7
SCHEMBL6533513 0.74 ALDH1A1 (0.44) ALDH1A1HPGDKDM4EIDO1HDAC8
Hydrochloric Acid SCHEMBL29287793 0.73 CA1 (0.47) ALDH1A1HPGDKDM4EBCAT2HSD17B10
SCHEMBL3701694 0.73 BCAT2 (0.46) ALDH1A1HPGDBCAT2HSD17B10USP2
Hydrochloric Acid SCHEMBL29287828 0.73 CA1 (0.47) ALDH1A1HPGDKDM4EBCAT2HSD17B10
SCHEMBL27647923 0.73 CDC7 (0.47) ALDH1A1KDM4ERPS6KB1CDC7ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed