SCHEMBL3714645

SCHEMBL3714645

CCOC(=O)c1csc(-c2ccc3[nH]ccc3c2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.60
RAB9A P51151 4/20 0.57
GAA P10253 1/20 0.57
NPC1 O15118 3/20 0.56
CLK1 P49759 1/20 0.56
MAPT P10636 3/20 0.51
POLB P06746 1/20 0.51
PKM P14618 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
ALDH1A1 P00352 3/20 0.49
CHEK1 O14757 2/20 0.48
CCNC P24863 1/20 0.46
CDK8 P49336 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
MAOA P21397 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
MMP2 P08253 1/20 0.44
MMP13 P45452 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3950463 0.80 EGFR (0.60) EGFRALDH1A1CHEK1CYP2C19GUSB
SCHEMBL7888746 0.80 RAB9A (0.53) EGFRRAB9AGAANPC1CLK1
SCHEMBL30443128 0.80 ACR (0.48) RAB9ANPC1MAPTPOLBALDH1A1
SCHEMBL3705300 0.80 RAB9A (0.50) EGFRRAB9AGAANPC1CLK1
SCHEMBL3702956 0.79 CDC7 (0.59) MAPTALDH1A1CCNCCDK8MEN1
SCHEMBL725782 0.79 MAOA (0.53) EGFRRAB9AGAANPC1MAPT
SCHEMBL27108838 0.79 RAB9A (0.72) RAB9AGAANPC1CLK1MAPT
SCHEMBL12582252 0.79 RAB9A (0.72) RAB9AGAANPC1CLK1MAPT
SCHEMBL3711151 0.78 CDC7 (0.59) EGFRCCNCCDK8MAOAMMP2
SCHEMBL18002724 0.78 RAB9A (0.61) RAB9AGAANPC1CLK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093191-A2 NOVEL COMPOUNDS EFFECTIVE AS XANTHINE OXIDASE INHIBITORS, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2010-08-19 WO disclosed
WO-2010093191-A2 NOVEL COMPOUNDS EFFECTIVE AS XANTHINE OXIDASE INHIBITORS, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2010-08-19 WO disclosed