SCHEMBL3715969

SCHEMBL3715969

CC(C)Oc1ccc(CCN(C#N)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.43
POLB P06746 1/20 0.43
KDM4E B2RXH2 1/20 0.41
NR1H4 Q96RI1 1/20 0.39
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSPO P30536 1/20 0.37
KMT2A Q03164 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
GLA P06280 1/20 0.36
HTR2A P28223 1/20 0.36
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PARP10 Q53GL7 1/20 0.35
ALPL P05186 1/20 0.35
ALPI P09923 1/20 0.35
ALPG P10696 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654575 0.82 CTSS (0.36) CTSSCTSK
SCHEMBL5170828 0.82 CTSS (0.48) KMT2ACTSSCTSKNPC1RAB9A
SCHEMBL3660898 0.74 MMP12 (0.51)
SCHEMBL3792997 0.73 GPR119 (0.46)
SCHEMBL8195571 0.71 CTSS (0.35) ALDH1A1CTSSCTSK
SCHEMBL7517658 0.70 ACACB (0.59) ACACBPOLBKDM4ENR1H4SMN1; SMN2
SCHEMBL12960637 0.70 POLB (0.68) ACACBPOLBKDM4ENR1H4ALDH1A1
SCHEMBL29101062 0.69 AOC3 (0.44) SMN1; SMN2KMT2ANPC1RAB9A
SCHEMBL2528423 0.69 RIPK1 (0.47) CTSSCTSK
SCHEMBL2809279 0.68 CTSK (0.48) ACACBPOLBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010108059-A1 SUBSTITUTED PYRIMIDINE DERIVATIVES AS ANTAGONISTS OF THE HISTAMINE H4 RECEPTOR INCYTE CORPORATION (US) 2010-09-23 WO disclosed