SCHEMBL3718669

SCHEMBL3718669

NCc1cc(-c2ccc(Br)cc2)nc(NCCc2ccc(S(N)(=O)=O)cc2)n1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 17/20 0.54
CA2 P00918 17/20 0.54
CA9 Q16790 16/20 0.54
CA12 O43570 4/20 0.53
CA14 Q9ULX7 2/20 0.53
CA4 P22748 2/20 0.53
CA3 P07451 1/20 0.53
CA6 P23280 1/20 0.53
CA7 P43166 1/20 0.53
CA13 Q8N1Q1 1/20 0.53
KDM4E B2RXH2 1/20 0.52
POLB P06746 1/20 0.52
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3717794 0.87 PTGS1 (0.54) CA1CA2CA9CA12CA14
SCHEMBL3718666 0.83 KDM4E (0.55) CA1CA2CA9CA12CA14
SCHEMBL3722029 0.77 L3MBTL1 (0.44) KDM4E
SCHEMBL3720119 0.75 ACP1 (0.44) KDM4E
SCHEMBL3723261 0.75 PTGS1 (0.48) CA1CA2CA9KDM4EPTGS1
SCHEMBL3720305 0.74 PIK3CA (0.43)
SCHEMBL3727322 0.71 AGTR1 (0.43) KDM4E
SCHEMBL3717789 0.71 SCN9A (0.53) CA1CA2CA9CA12CA14
SCHEMBL3723029 0.69 KDM4E (0.53) KDM4E
SCHEMBL3717784 0.69 ACP1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed