SCHEMBL3718696

SCHEMBL3718696

CC(C)c1n[nH]c2c(NCc3cc(F)ccc3O)nc(NCCCN)nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 10/20 0.43
CCNE1 P24864 9/20 0.43
CCNT1 O60563 4/20 0.43
CDK9 P50750 4/20 0.43
CDK5 Q00535 4/20 0.43
CDK5R1 Q15078 3/20 0.43
CDK7 P50613 2/20 0.43
CCNH P51946 2/20 0.43
CCNE2 O96020 4/20 0.41
CCNT2 O60583 2/20 0.41
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
BCDIN3D Q7Z5W3 1/20 0.37
CCNA2 P20248 2/20 0.37
CCNA1 P78396 2/20 0.37
MAP2K4 P45985 1/20 0.35
TACR2 P21452 1/20 0.35
NTRK1 P04629 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724487 0.89 CDK2 (0.47) CDK2CCNE1CCNT1CDK9CDK5
SCHEMBL3722170 0.87 CCNE1 (0.44) CDK2CCNE1CCNT1CDK9CDK5
SCHEMBL3725653 0.86 CDK2 (0.46) CDK2CCNE1CDK5CCNE2CCNB2
SCHEMBL3720124 0.86 CCNE1 (0.43) CDK2CCNE1CCNT1CDK9CDK5
SCHEMBL3718690 0.85 CDK2 (0.51) CDK2CCNE1CCNT1CDK9CDK5
SCHEMBL3724956 0.84 CDK2 (0.42) CDK2CCNE1CCNT1CDK9CDK5
SCHEMBL3716187 0.84 CDK2 (0.43) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3721963 0.83 P2RX7 (0.41) CDK2CCNE1CDK5CCNE2CCNB2
SCHEMBL3724809 0.83 CDK2 (0.40) CDK2CCNE1CDK5CDK7CCNE2
SCHEMBL3718378 0.82 CDK2 (0.43) CDK2CCNE1CCNT1CDK9CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139288-A1 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS C3 BIO GMBH (DE) 2010-12-09 WO disclosed