SCHEMBL3720892

SCHEMBL3720892

CCC(C(=O)O)c1ccc(Oc2ccc3cc(CCN)ccc3n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.46
AKR1C2 P52895 8/20 0.46
AKR1C1 Q04828 1/20 0.46
PTGS1 P23219 1/20 0.46
SCN9A Q15858 9/20 0.39
F2 P00734 1/20 0.39
SCN10A Q9Y5Y9 2/20 0.38
PDE4B Q07343 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721946 0.87 SCN9A (0.40) AKR1C3AKR1C2AKR1C1PTGS1SCN9A
SCHEMBL3720891 0.84 AKR1C3 (0.51) AKR1C3AKR1C2AKR1C1PTGS1SCN9A
SCHEMBL3721431 0.82 PDE4B (0.53) AKR1C3AKR1C2AKR1C1PTGS1SCN9A
SCHEMBL3726204 0.81 LOXL2 (0.49) SCN9AF2PDE4B
SCHEMBL3717827 0.80 ALDH1A1 (0.49)
SCHEMBL3720365 0.78 MAPT (0.41)
SCHEMBL3717202 0.78 ACACB (0.38)
SCHEMBL3717681 0.78 HTT (0.49)
SCHEMBL3722365 0.77 ALOX5 (0.38) SCN9ASCN10A
SCHEMBL3720293 0.77 GLA (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed