SCHEMBL3723608

SCHEMBL3723608

Cc1nn(C2CCOCC2)c(N2CCCC2C(=O)O)c1S(=O)(=O)c1ccc(OCC(F)(F)F)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.38
CTSS P25774 5/20 0.37
PPARG P37231 2/20 0.33
PPARD Q03181 2/20 0.33
PPARA Q07869 2/20 0.33
CTSL P07711 2/20 0.33
PRCP P42785 1/20 0.33
AOC2 O75106 1/20 0.33
MAOA P21397 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
P2RX7 Q99572 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
HSD11B1 P28845 1/20 0.32
KCNJ6 P48051 1/20 0.32
KCNJ5 P48544 1/20 0.32
KCNJ3 P48549 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718383 0.89 CTSS (0.36) RORCCTSSAOC2MAOAP2RX7
SCHEMBL3725935 0.86 P2RX7 (0.43) RORCP2RX7HSD11B1
SCHEMBL3719493 0.83 CTSS (0.37) RORCCTSSHSD11B1
SCHEMBL697204 0.82 KEAP1 (0.37) RORCHCRTR1HCRTR2
SCHEMBL690481 0.82 TSHR (0.36) CTSSP2RX7HSD11B1
SCHEMBL696119 0.81 HSD11B1 (0.41) RORCCTSSCTSLP2RX7HSD11B1
SCHEMBL694889 0.79 P2RX7 (0.40) RORCCTSSCTSLP2RX7HCRTR1
SCHEMBL3719407 0.78 CFTR (0.36) RORCHSD11B1
SCHEMBL695720 0.76 CTSS (0.37) CTSSP2RX7HSD11B1KCNJ6KCNJ5
SCHEMBL694457 0.76 AADAT (0.36) CTSSITGB1ITGA4HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed