SCHEMBL3725935

SCHEMBL3725935

Cc1nn(C2CCOCC2)c(N2CCCC2C(=O)O)c1S(=O)(=O)c1ccc(F)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.43
MAPT P10636 2/20 0.35
CFTR P13569 2/20 0.34
RORC P51449 1/20 0.34
EPHX2 P34913 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
AGTR2 P50052 2/20 0.33
PDE9A O76083 1/20 0.33
HSD11B1 P28845 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL694889 0.93 P2RX7 (0.40) P2RX7MAPTRORCEPHX2HSD11B1
SCHEMBL696119 0.89 HSD11B1 (0.41) P2RX7CFTRRORCEPHX2KDM4C
SCHEMBL690481 0.88 TSHR (0.36) P2RX7MAPTCFTRHSD11B1KMT2A
SCHEMBL3723608 0.86 RORC (0.38) P2RX7RORCHSD11B1
SCHEMBL3718383 0.85 CTSS (0.36) P2RX7RORCHSD11B1KMT2A
SCHEMBL696084 0.84 P2RX7 (0.40) P2RX7EPHX2
SCHEMBL697204 0.82 KEAP1 (0.37) RORCAGTR2
SCHEMBL694457 0.81 AADAT (0.36) MAPTHSD11B1
SCHEMBL697628 0.80 CTSL (0.38) P2RX7RORCEPHX2HSD11B1
SCHEMBL696136 0.80 AADAT (0.39) MAPTHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed