SCHEMBL3727020

SCHEMBL3727020

CS(=O)(=O)c1ccc(-c2cccc(CN)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 1/20 0.55
NMT1 P30419 1/20 0.54
CA12 O43570 3/20 0.49
CA2 P00918 3/20 0.49
CA9 Q16790 3/20 0.49
USP28 Q96RU2 1/20 0.47
PTGS2 P35354 4/20 0.47
TAAR1 Q96RJ0 3/20 0.46
PSIP1 O75475 1/20 0.44
PTGS1 P23219 1/20 0.44
CA1 P00915 2/20 0.44
RORC P51449 1/20 0.43
KIF11 P52732 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
FYN P06241 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3655415 0.88 LOXL2 (0.54) ADAMTS4NMT1USP28PSIP1KIF11
SCHEMBL4183608 0.86 PSIP1 (0.59) CA12CA2CA9USP28PTGS2
SCHEMBL3720559 0.85 CA2 (0.70) ADAMTS4NMT1CA12CA2CA9
SCHEMBL13675350 0.85 BCL2 (0.57) CA12CA2CA9PTGS2PTGS1
Hydrochloric Acid SCHEMBL4199854 0.84 CA1 (0.59) CA12CA2CA9USP28PTGS2
SCHEMBL2025954 0.83 FYN (0.57) ADAMTS4CA12CA2CA9PTGS2
SCHEMBL19496815 0.81 HSD17B1 (0.53) NMT1PTGS2TAAR1RORC
SCHEMBL1127911 0.80 HTR6 (0.51) CA12CA2CA9USP28PSIP1
SCHEMBL201356 0.80 PSIP1 (0.65) CA12CA2CA9PTGS2PSIP1
SCHEMBL3794460 0.80 TAAR1 (0.70) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed