SCHEMBL3727231

SCHEMBL3727231

N#Cc1ccc(-c2cc(CN)nc(N3CCN(c4ccccc4F)CC3)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 3/20 0.42
ATM Q13315 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
HRH4 Q9H3N8 3/20 0.41
HRH3 Q9Y5N1 2/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2C P18825 1/20 0.40
HTR1D P28221 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR7 P34969 1/20 0.40
MAPT P10636 3/20 0.39
HTT P42858 2/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720242 0.90 HRH4 (0.46) ALDH1A1KMT2AKDM4EATMSMN1; SMN2
SCHEMBL3727042 0.88 DRD2 (0.47) ALDH1A1KDM4ESMN1; SMN2NPC1LMNA
SCHEMBL3718590 0.88 ALDH1A1 (0.52) ALDH1A1KMT2AKDM4EATMSMN1; SMN2
SCHEMBL3721161 0.86 MAPT (0.44) ALDH1A1KMT2ASMN1; SMN2NPC1LMNA
SCHEMBL3721032 0.84 CYP1A2 (0.44) ALDH1A1KMT2AKDM4EATMSMN1; SMN2
SCHEMBL3721047 0.84 SMN1; SMN2 (0.45) ALDH1A1KMT2AKDM4ESMN1; SMN2NPC1
SCHEMBL3724712 0.82 LMNA (0.42) ALDH1A1KDM4ESMN1; SMN2NPC1LMNA
SCHEMBL3717916 0.82 LMNA (0.42) ALDH1A1KDM4ESMN1; SMN2NPC1LMNA
SCHEMBL3721778 0.82 SMN1; SMN2 (0.46) ALDH1A1KMT2AKDM4ESMN1; SMN2NPC1
SCHEMBL3722201 0.82 ALDH1A1 (0.46) ALDH1A1KMT2AKDM4ESMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed