SCHEMBL374569

SCHEMBL374569

Nc1ccc(OCCCN2CCOCC2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.74
MAPK1 P28482 2/20 0.74
ALDH1A1 P00352 1/20 0.74
CYP1A2 P05177 1/20 0.74
CHRM2 P08172 1/20 0.74
CHRM1 P11229 1/20 0.74
HTR2A P28223 1/20 0.74
SCN1A P35498 1/20 0.74
HTR2B P41595 1/20 0.74
KCNH2 Q12809 1/20 0.74
SCN2A Q99250 1/20 0.74
SIGMAR1 Q99720 1/20 0.74
SCN3A Q9NY46 1/20 0.74
USP2 O75604 1/20 0.72
LMNA P02545 1/20 0.72
HRH2 P25021 1/20 0.63
HRH1 P35367 1/20 0.63
TSHR P16473 1/20 0.60
CA12 O43570 1/20 0.57
CA1 P00915 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14724514 0.95 HRH3 (0.71) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL28126773 0.95 HRH3 (0.68) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL16314572 0.94 ALDH1A1 (0.66) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL18763519 0.93 HRH3 (0.65) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL374497 0.92 LTA4H (0.67) HRH3MAPK1ALDH1A1CYP1A2CHRM2
Hydrochloric Acid SCHEMBL2385707 0.90 NPC1 (0.68) HRH3MAPK1ALDH1A1CYP1A2CHRM2
Hydrochloric Acid SCHEMBL14742325 0.90 NPC1 (0.68) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL14204158 0.90 CA12 (0.65) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL24398699 0.89 TSHR (0.76) HRH3MAPK1ALDH1A1CYP1A2CHRM2
SCHEMBL22609310 0.89 LTA4H (0.65) HRH3MAPK1ALDH1A1CYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 108 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4673149-A1 NEW COMPOUNDS AND TREATMENT OF RENAL CELL CARCINOMA Trustlife Global Inc. (US) 2026-01-07 EP disclosed
US-20250188041-A1 NEW COMPOUNDS AND TREATMENT OF RENAL CELL CARCINOMA Trustlife Global Inc. 2025-06-12 US disclosed
EP-4486348-A1 NEW COMPOUNDS AND TREATMENT OF RENAL CELL CARCINOMA Trustlife Global Inc. (US) 2025-01-08 EP disclosed
CN-118804751-A New compounds and treatment of renal cell carcinoma 巴什生物技术公司 2024-10-18 CN disclosed
CN-116120300-B Pyrimidine compound containing hydroxamic acid fragment, and preparation method and application thereof 贵州大学 2024-10-15 CN disclosed
WO-2024179699-A1 NEW COMPOUNDS AND TREATMENT OF RENAL CELL CARCINOMA BASH BIOTECH INC. (US) 2024-09-06 WO disclosed
CN-114716366-B 3-hydroxypyridin-4-one derivatives and application thereof in inhibiting iron death of renal cells 浙江大学 2023-12-26 CN disclosed
WO-2023166153-A1 NEW COMPOUNDS AND TREATMENT OF RENAL CELL CARCINOMA BASH BIOTECH INC (US) 2023-09-07 WO disclosed
CN-116120300-A Pyrimidine compound containing hydroxamic acid fragment, and preparation method and application thereof 贵州大学 2023-05-16 CN disclosed
US-11007193-B2 2,4-pyrimidinediamine compounds and their uses RIGEL PHARMACEUTICALS, INC. (US) 2021-05-18 US disclosed
US-20070293524-A1 Salts, hydrates, solvatesand/or N-oxides; inhibit the IgE and/or IgG receptor signaling cascades that lead to the release of chemical mediators; Syk kinase inhibitors; inhibiting an Fc receptor signal transduction cascade RIGEL PHARMACEUTICALS, INC. (US) 2007-12-20 US disclosed
US-20070225321-A1 2,4-PYRIMIDINEDIAMINE COMPOUNDS AND THEIR USES RIGEL PHARMACEUTICALS, INC. (US) 2007-09-27 US disclosed
EP-1761505-A1 PYRIMIDINE UREA DERIVATIVES AS KINASE INHIBITORS Novartis AG (CH) 2007-03-14 EP disclosed
WO-2007018941-A2 PYRIMIDYL-THIOPHENE DERIVATIVES SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed
US-7060827-B2 Prevent immunoglobulin receptors signaling cascading; prevention diseases; drugs; antiinflammatory agents RIGEL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
WO-2006000420-A1 PYRIMIDINE UREA DERIVATIVES AS KINASE INHIBITORS NOVARTIS AG (CH) 2006-01-05 WO disclosed
CN-1678321-A Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds RIGEL PHARMACEUTICALS INC (US) 2005-10-05 CN disclosed
US-20050209230-A1 2-leaving group-4-(substituted amino)-5-fluoropyrimidines such as 2-chloro-N4-(2-hydroxyphenyl)-5-fluoro-4-pyrimidineamine; chemical intermediates to compounds that inhibit the immunoglobulin (Ig) IgE and/or IgG receptor signaling cascades MIDCAP FINANCIAL TRUST 2005-09-22 US disclosed
US-20050038243-A1 Prevent immunoglobulin receptors signaling cascading; prevention diseases; drugs; antiinflammatory agents MIDCAP FINANCIAL TRUST 2005-02-17 US disclosed
US-20040029902-A1 Antiinflamamtory agents MIDCAP FINANCIAL TRUST 2004-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070225321-A1 2,4-PYRIMIDINEDIAMINE COMPOUNDS AND THEIR USES FCER2, FCGR1A, FCGR2A HRH3 22/4885MAPK1 581/4885ALDH1A1 2891/4885
US-20040029902-A1 Antiinflamamtory agents FCER2, FCGR1A, HNMT HRH3 25/4885MAPK1 1201/4885ALDH1A1 2723/4885
US-20050209230-A1 2-leaving group-4-(substituted amino)-5-fluoropyrimidines such as 2-chloro-N4-(2-hydroxyphenyl)-5-fluoro-4-pyrimidineamine; chemical intermediates to compounds that inhibit the immunoglobulin (Ig) IgE and/or IgG receptor signaling cascades FCER2, FCGR1A, FCGR2A HRH3 16/4885MAPK1 1247/4885ALDH1A1 2615/4885
US-20050038243-A1 Prevent immunoglobulin receptors signaling cascading; prevention diseases; drugs; antiinflammatory agents FCER2, FCGR1A, FCGR2A HRH3 131/4885MAPK1 434/4885ALDH1A1 2302/4885
US-20250188041-A1 NEW COMPOUNDS AND TREATMENT OF RENAL CELL CARCINOMA RCC2, GLS, VHL HRH3 3810/4885MAPK1 1240/4885ALDH1A1 208/4885
US-11007193-B2 2,4-pyrimidinediamine compounds and their uses FCER2, FCGR1A, FCGR2A HRH3 22/4885MAPK1 581/4885ALDH1A1 2891/4885
US-20070293524-A1 Salts, hydrates, solvatesand/or N-oxides; inhibit the IgE and/or IgG receptor signaling cascades that lead to the release of chemical mediators; Syk kinase inhibitors; inhibiting an Fc receptor signal transduction cascade SYK, FCER2, FCGR1A HRH3 65/4885MAPK1 233/4885ALDH1A1 3950/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.