SCHEMBL3753543

SCHEMBL3753543

O=C(C(=O)c1ccc(C#Cc2ccc(C(F)(F)F)cc2)cc1)c1ccc(C#Cc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.76
CES1 P23141 2/20 0.76
RARB P10826 1/20 0.50
RARG P13631 1/20 0.50
SRD5A2 P31213 1/20 0.50
PTPN1 P18031 3/20 0.48
GSK3B P49841 2/20 0.48
NR4A1 P22736 1/20 0.44
NR4A2 P43354 1/20 0.44
NR4A3 Q92570 1/20 0.44
MEN1 O00255 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
PTPN6 P29350 1/20 0.43
PTPN11 Q06124 1/20 0.43
KIF11 P52732 1/20 0.42
EPHX2 P34913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3172262 0.87 CES2 (1.00) CES2CES1SRD5A2PTPN1GSK3B
SCHEMBL22721378 0.86 SRD5A2 (0.69) CES2CES1RARBRARGSRD5A2
SCHEMBL22721407 0.85 MAOB (0.58) CES2CES1RARBRARGSRD5A2
SCHEMBL14998069 0.82 KIF11 (0.56) CES2CES1TSHRKIF11
SCHEMBL16747679 0.82 KIF11 (0.56) CES2CES1TSHRKIF11
SCHEMBL9876492 0.80 PTPN11 (0.55) CES2CES1RARBRARGPTPN11
SCHEMBL17191457 0.80 RARB (0.76) CES2CES1RARBRARGSRD5A2
SCHEMBL20010796 0.79 CES2 (0.83) CES2CES1SRD5A2PTPN1GSK3B
SCHEMBL2834217 0.79 CES2 (0.83) CES2CES1SRD5A2PTPN1GSK3B
SCHEMBL3753473 0.78 CES2 (0.45) CES2CES1RARBRARGSRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7842830-B2 Transition-metal charge-transport materials, methods of fabrication thereof, and methods of use thereof GEORGIA TECH RESEARCH CORPORATION (US) 2010-11-30 US disclosed
US-20080121870-A1 Transition-Metal Charge Transport Materials, Methods Of Fabrication Thereof, And Methods Of Use Thereof GEORGIA TECH RESEACH CORPORATION 2008-05-29 US disclosed
WO-2005123754-A2 TRANSITION-METAL CHARGE-TRANSPORT MATERIALS, METHODS OF FABRICATION THEREOF, AND METHODS OF USE THEREOF GEORGIA TECH RESEARCH CORPORATION (US) 2005-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080121870-A1 Transition-Metal Charge Transport Materials, Methods Of Fabrication Thereof, And Methods Of Use Thereof SLC39A3, SLC6A6, SLC6A9 CES2 1387/4885CES1 4295/4885RARB 3210/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.