SCHEMBL3763934

SCHEMBL3763934

CC(C)(C)OC(=O)NCC(=O)N1CCC[C@H]1C(N)=O

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TSHR P16473 1/20 0.48
KMT2A Q03164 1/20 0.48
DPP4 P27487 8/20 0.43
FAP Q12884 4/20 0.43
PREP P48147 2/20 0.43
ACE P12821 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KLK5 Q9Y337 1/20 0.41
MMP1 P03956 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2744394 1.00 MEN1 (0.48) MEN1ALDH1A1TSHRKMT2ADPP4
SCHEMBL13580680 0.90 MEN1 (0.43) MEN1ALDH1A1TSHRKMT2ADPP4
SCHEMBL1000948 0.88 ACE (0.53) MEN1ALDH1A1TSHRKMT2AFAP
SCHEMBL8352289 0.88 MEN1 (0.49) MEN1ALDH1A1TSHRKMT2ADPP4
SCHEMBL14979025 0.88 MEN1 (0.49) MEN1ALDH1A1TSHRKMT2ADPP4
SCHEMBL1925210 0.88 ACE (0.53) MEN1ALDH1A1TSHRKMT2AFAP
SCHEMBL8131025 0.88 DPP4 (0.43) MEN1ALDH1A1TSHRKMT2ADPP4
SCHEMBL10881232 0.87 DPP4 (0.49) DPP4ACESMN1; SMN2KLK5
SCHEMBL6468703 0.87 KLK5 (0.53) MEN1ALDH1A1TSHRKMT2ADPP4
SCHEMBL14235217 0.87 KLK5 (0.53) MEN1ALDH1A1TSHRKMT2ADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025237891-A1 QUINOLINE-2-CARBOXAMIDE DERIVATIVES AS RAD51 INHIBITORS FOR THE TREATMENT OF CANCER NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2025-11-20 WO disclosed
US-20250235566-A1 TRISLINKER-CONJUGATED DIMERIC LABELING PRECURSORS AND RADIOTRACERS DERIVED THEREFROM Medianezia GmbH (DE) 2025-07-24 US disclosed
EP-4351663-A1 TRISLINKER-CONJUGATED DIMERIC LABELLING PRECURSORS AND RADIOTRACERS DERIVED THEREFROM Medianezia GmbH (DE) 2024-04-17 EP disclosed
US-11858924-B2 N-(2-(4-cyanothiazolidin-3-yl)-2-oxoethyl)-quinoline-4-carboxamides ASTRAZENECA (SE) 2024-01-02 US disclosed
US-20230312550-A1 N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-QUINOLINE-4-CARBOXAMIDES ASTRAZENECA AB (SE) 2023-10-05 US disclosed
WO-2022258637-A1 TRISLINKER-CONJUGATED DIMERIC LABELLING PRECURSORS AND RADIOTRACERS DERIVED THEREFROM Atoms for Cure GmbH (DE) 2022-12-15 WO disclosed
US-20210369877-A1 MARKING PRECURSOR WITH SQUARIC ACID COUPLING SCV- Spezial Chemikalien Vertrieb GmbH (DE) 2021-12-02 US disclosed
EP-2804859-B1 NOVEL FAP INHIBITORS UNIV ANTWERPEN (BE) 2019-06-12 EP disclosed
EP-2246347-B1 DICYCLOAZAALKANE DERIVATES, PREPARATION PROCESSES AND MEDICAL USES THEREOF SHANGHAI HENGRUI PHARM CO LTD (CN) 2016-09-28 EP disclosed
US-9346814-B2 FAP inhibitors Universiteit Antwerp (BE) 2016-05-24 US disclosed
US-20100311747-A1 DICYCLOAZAALKANE DERIVATES, PREPARATION PROCESSES AND MEDICAL USES THEREOF SHANGHAI HENGRUI PHARMACEUTICAL CO. LTD. (CN) 2010-12-09 US disclosed
US-20100311747-A1 DICYCLOAZAALKANE DERIVATES, PREPARATION PROCESSES AND MEDICAL USES THEREOF SHANGHAI HENGRUI PHARMACEUTICAL CO. LTD. (CN) 2010-12-09 US disclosed
WO-2009142842-A9 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2010-11-25 WO disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed
US-20090176847-A1 Dicyclooctane Derivatives, Preparation Processes and Medical Uses Thereof SHANGHAI HENGRUI PHARMACEUTICAL CO., LTD. (CN) 2009-07-09 US disclosed
US-20090176847-A1 Dicyclooctane Derivatives, Preparation Processes and Medical Uses Thereof SHANGHAI HENGRUI PHARMACEUTICAL CO., LTD. (CN) 2009-07-09 US disclosed
WO-2009005677-A2 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2009-01-08 WO disclosed
EP-2006284-A1 DICYCLOOCTANE DERIVATES, PREPARATION PROCESSES AND MEDICAL USES THEREOF Shanghai Hengrui Pharmaceutical Co. Ltd. (CN) 2008-12-24 EP disclosed
WO-2008137779-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2008-11-13 WO disclosed
WO-2007015824-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2007-02-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176847-A1 Dicyclooctane Derivatives, Preparation Processes and Medical Uses Thereof DPP4, DPP7, DPP8 MEN1 1501/4885ALDH1A1 1142/4885TSHR 4125/4885
US-20100311747-A1 DICYCLOAZAALKANE DERIVATES, PREPARATION PROCESSES AND MEDICAL USES THEREOF DPP4, DPP8, DPP7 MEN1 2775/4885ALDH1A1 451/4885TSHR 3534/4885
US-20250235566-A1 TRISLINKER-CONJUGATED DIMERIC LABELING PRECURSORS AND RADIOTRACERS DERIVED THEREFROM TK1, TK2, TMT1A MEN1 385/4885ALDH1A1 2879/4885TSHR 81/4885
US-20230312550-A1 N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-QUINOLINE-4-CARBOXAMIDES FAP, PREP, CTRL MEN1 1482/4885ALDH1A1 1593/4885TSHR 1989/4885
US-20210369877-A1 MARKING PRECURSOR WITH SQUARIC ACID COUPLING SCLY, SRRT, CS MEN1 2064/4885ALDH1A1 1074/4885TSHR 162/4885
US-11858924-B2 N-(2-(4-cyanothiazolidin-3-yl)-2-oxoethyl)-quinoline-4-carboxamides FAP, PREP, CTRL MEN1 1482/4885ALDH1A1 1593/4885TSHR 1989/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.