SCHEMBL377104

SCHEMBL377104

OB(O)c1cccnc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MMP2 P08253 2/20 0.37
TSHR P16473 2/20 0.37
CHRM1 P11229 1/20 0.37
COMT P21964 1/20 0.37
ADRA1A P35348 1/20 0.37
METAP2 P50579 1/20 0.37
METAP1 P53582 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HTT P42858 2/20 0.36
SLC6A2 P23975 1/20 0.36
LIPE Q05469 1/20 0.35
HSP90AA1 P07900 3/20 0.34
NPC1 O15118 2/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29823712 1.00 ENPP2 (0.38) ENPP2L3MBTL1ALDH1A1MMP2TSHR
SCHEMBL29515564 0.78 P2RX7 (0.41) ENPP2L3MBTL1ALDH1A1HTTSLC6A2
SCHEMBL29232877 0.78 ENPP2 (0.37) ENPP2L3MBTL1MMP2TSHRHTT
SCHEMBL586439 0.78 P2RX7 (0.41) ENPP2L3MBTL1ALDH1A1HTTSLC6A2
SCHEMBL28165 0.76 NAPRT (0.45) ENPP2L3MBTL1LIPEHSP90AA1NPC1
SCHEMBL29952309 0.76 NOS3 (0.52) ENPP2ALDH1A1HSP90AA1NOS3NOS1
SCHEMBL1920925 0.76 TRIM24 (0.47) ENPP2L3MBTL1HTTLIPEHSP90AA1
SCHEMBL117563 0.76 NOS3 (0.52) ENPP2ALDH1A1HSP90AA1NOS3NOS1
Hydrochloric Acid SCHEMBL14797461 0.76 P2RX7 (0.40) ENPP2L3MBTL1ALDH1A1HTTSLC6A2
SCHEMBL315754 0.76 SMN1; SMN2 (0.45) ENPP2ALDH1A1HTTNPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 84 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12421273-B2 Ectonucleotidase inhibitors and methods of use thereof ANTENGENE THERAPEUTICS LIMITED (CN) 2025-09-23 US disclosed
US-20250206757-A1 5,8-DIHYDRO-1,7-NAPHTHYRIDINE DERIVATIVES AS GLP-1 AGONISTS FOR THE TREATMENT OF DIABETES GASHERBRUM BIO, INC. 2025-06-26 US disclosed
US-12297208-B2 Small molecule inhibitors of KRAS G12C mutant MERCK SHARP & DOHME LLC (US) 2025-05-13 US disclosed
US-12291538-B2 Small molecule inhibitors of KRAS G12C mutant MERCK SHARP & DOHME LLC (US) 2025-05-06 US disclosed
EP-4496797-A1 5,8-DIHYDRO-1,7-NAPHTHYRIDINE DERIVATIVES AS GLP-1 AGONISTS FOR THE TREATMENT OF DIABETES Gasherbrum Bio, Inc. (US) 2025-01-29 EP disclosed
CN-118359538-A Isoquinoline compound, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2024-07-19 CN disclosed
US-20240132533-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF ANTENGENT THERAPEUTICS LIMITED (CN) 2024-04-25 US disclosed
CN-112888696-B Exonuclease inhibitors and methods of use thereof 德琪医疗有限公司 2024-04-16 CN disclosed
US-20240092744-A1 TRICYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF THE NATIONAL INSTITUTES OF PHARMACEUTICAL R&D CO., LTD (CN) 2024-03-21 US disclosed
US-20240083913-A1 Small Molecule Inhibitors of KRAS G12C Mutant MERCK SHARP & DOHME LLC 2024-03-14 US disclosed
US-20110033417-A1 2,3-SUBSTITUTED INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS MERCK SHARP & DOHME CORP. 2011-02-10 US disclosed
US-20100239527-A1 2,3-SUBSTITUTED AZAINDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS SCHERING CORPORATION (US) 2010-09-23 US disclosed
EP-2197842-A1 2, 3-SUBSTITUTED INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS SCHERING CORPORATION (US) 2010-06-23 EP disclosed
EP-2195317-A1 2,3-SUBSTITUTED AZAINDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS SCHERING CORPORATION (US) 2010-06-16 EP disclosed
US-20100098661-A1 4,5-RING ANNULATED INDOLE DERIVATIVES FOR TREATING OR PREVENTING OF HCV AND RELATED VIRAL INFECTIONS SCHERING CORPORATION 2010-04-22 US disclosed
EP-2064180-A1 4,5-RING ANNULATED INDOLE DERIVATIVES FOR TREATING OR PREVENTING OF HCV AND RELATED VIRAL INFECTIONS SCHERING CORPORATION (US) 2009-06-03 EP disclosed
WO-2009032125-A1 2,3-SUBSTITUTED AZAINDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS SCHERING CORPORATION (US) 2009-03-12 WO disclosed
WO-2009032116-A1 2, 3-SUBSTITUTED INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS SCHERING CORPORATION (US) 2009-03-12 WO disclosed
WO-2009032124-A1 SUBSTITUTED INDOLE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION (US) 2009-03-12 WO disclosed
WO-2008082484-A1 4,5-RING ANNULATED INDOLE DERIVATIVES FOR TREATING OR PREVENTING OF HCV AND RELATED VIRAL INFECTIONS SCHERING CORPORATION (US) 2008-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240132533-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF NT5E, ENTPD5, NT5C2 ENPP2 17/4885L3MBTL1 4683/4885ALDH1A1 527/4885
US-20110033417-A1 2,3-SUBSTITUTED INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS IDO2, IDO1, IRF3 ENPP2 1483/4885L3MBTL1 995/4885ALDH1A1 1792/4885
US-12297208-B2 Small molecule inhibitors of KRAS G12C mutant KRAS, NRAS, HRAS ENPP2 3262/4885L3MBTL1 1874/4885ALDH1A1 4287/4885
US-12421273-B2 Ectonucleotidase inhibitors and methods of use thereof NT5E, ENTPD5, NT5C2 ENPP2 17/4885L3MBTL1 4683/4885ALDH1A1 527/4885
US-20100098661-A1 4,5-RING ANNULATED INDOLE DERIVATIVES FOR TREATING OR PREVENTING OF HCV AND RELATED VIRAL INFECTIONS ZC3HAV1, IDO1, ZC3HAV1L ENPP2 2861/4885L3MBTL1 2367/4885ALDH1A1 248/4885
US-20240092744-A1 TRICYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF GOT2, HADH, CYP4A11 ENPP2 2038/4885L3MBTL1 1801/4885ALDH1A1 52/4885
US-20250206757-A1 5,8-DIHYDRO-1,7-NAPHTHYRIDINE DERIVATIVES AS GLP-1 AGONISTS FOR THE TREATMENT OF DIABETES GLP1R, IAPP, GPR119 ENPP2 298/4885L3MBTL1 3471/4885ALDH1A1 1791/4885
US-20240083913-A1 Small Molecule Inhibitors of KRAS G12C Mutant KRAS, NRAS, HRAS ENPP2 3262/4885L3MBTL1 1874/4885ALDH1A1 4287/4885
US-12291538-B2 Small molecule inhibitors of KRAS G12C mutant KRAS, NRAS, HRAS ENPP2 3262/4885L3MBTL1 1874/4885ALDH1A1 4287/4885
US-20100239527-A1 2,3-SUBSTITUTED AZAINDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS HAVCR2, AZI2, ZC3HAV1 ENPP2 795/4885L3MBTL1 1514/4885ALDH1A1 1912/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.