SCHEMBL3772998

SCHEMBL3772998

CC(C)(C)OC(=O)N=C(N)N(C(=O)OC(C)(C)C)c1ccc2c(c1)CCC2

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 1/20 0.38
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
NR1H2 P55055 1/20 0.33
ALDH1A1 P00352 1/20 0.32
ESR2 Q92731 1/20 0.32
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3784231 0.88 MT-CO2 (0.31) MT-CO2NR1H2
SCHEMBL3778075 0.81 TP53 (0.31)
SCHEMBL17894521 0.79 MIF (0.36) MT-CO2
SCHEMBL3777967 0.79 SCN2A (0.32) MT-CO2ALDH1A1
SCHEMBL3785117 0.77 KMT2A (0.34) RAB9AALDH1A1
SCHEMBL15876020 0.77 MAPT (0.39) NPC1RXRARXRBRXRGALDH1A1
SCHEMBL3775825 0.76 KDM4E (0.33) NPC1RAB9AALDH1A1
SCHEMBL15140038 0.75 F2 (0.35) NPC1RAB9ARXRARXRBALDH1A1
SCHEMBL207903 0.74 MTNR1B (0.35) NR1H2
SCHEMBL7797012 0.74 UNG (0.32) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100331384-A1 GUANIDINE BASED COMPOUNDS UNIVERSIDAD DEL PAIS VASCO/EUSKAL HERRIKO UNIBERTSITATEA (ES) 2010-12-30 US disclosed
WO-2009080818-A2 GUANIDINE BASED COMPOUNDS THE PROVOST, FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2009-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100331384-A1 GUANIDINE BASED COMPOUNDS ADRB2, ADRA2A, ADRA2C MT-CO2 2178/4885NPC1 3544/4885RAB9A 648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.