SCHEMBL3785370

SCHEMBL3785370

CC(=O)C(Cc1ccc(Cl)cc1)C(=O)Nc1cc(O)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LNPEP Q9UIQ6 3/20 0.40
ERAP2 Q6P179 2/20 0.40
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PPARG P37231 2/20 0.38
PPARA Q07869 2/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
NLRP3 Q96P20 1/20 0.37
GPR142 Q7Z601 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
TMPRSS4 Q9NRS4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3784633 0.91 GAA (0.42) MDM2MEN1KMT2ALNPEPERAP2
SCHEMBL2577121 0.89 LNPEP (0.39) MEN1KMT2AL3MBTL1LNPEPERAP2
SCHEMBL3784324 0.89 MEN1 (0.53) MEN1KMT2AL3MBTL1LNPEPERAP2
SCHEMBL534032 0.86 GPR142 (0.39) LNPEPERAP2NLRP3GPR142TMPRSS4
SCHEMBL3779263 0.86 ALDH1A1 (0.38) MEN1KMT2AL3MBTL1LNPEPERAP2
SCHEMBL3779106 0.86 ANO1 (0.37) MEN1KMT2AALDH1A1KDM4ESMN1; SMN2
SCHEMBL2581345 0.85 LNPEP (0.41) MDM2LNPEPERAP2ALDH1A1PPARG
SCHEMBL3783304 0.85 KIF11 (0.41) L3MBTL1LNPEPERAP2ALDH1A1
SCHEMBL3772879 0.85 HDAC8 (0.43) MEN1KMT2AALDH1A1KDM4E
SCHEMBL3775842 0.81 PYGL (0.41) MDM2MEN1KMT2AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7858640-B2 Quinolines and their therapeutic use PULMAGEN THERAPEUTICS (ASTHMA) LIMITED (GB) 2010-12-28 US disclosed
US-20090156600-A1 Quinolines and Their Therapeutic Use GB005, INC. 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156600-A1 Quinolines and Their Therapeutic Use NR3C1, NR3C2, NR1H3 MDM2 4600/4885MEN1 4140/4885KMT2A 3406/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.