Water

Water

SCHEMBL3820520

O.O.O.O.O.O.O.[KH]

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL9484116 1.00
Water SCHEMBL8369534 1.00
Water SCHEMBL1504321 1.00
Water SCHEMBL8466165 1.00
Water SCHEMBL22588912 1.00
Water SCHEMBL1530181 1.00
Water SCHEMBL8193216 1.00
Water SCHEMBL6228132 1.00
Water SCHEMBL3819207 1.00
Water SCHEMBL797313 1.00

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478339-B9 PHARMACEUTICAL FORMULATIONS OF ANTINEOPLASTIC AGENTS, IN PARTICULAR TEMOZOLOMIDE, PROCESSES OF MAKING AND USING THE SAME SCHERING CORP (US) 2009-08-19 EP claimed
EP-1478339-B1 PHARMACEUTICAL FORMULATIONS OF ANTINEOPLASTIC AGENTS, IN PARTICULAR TEMOZOLOMIDE, PROCESSES OF MAKING AND USING THE SAME SCHERING CORP (US) 2008-06-04 EP claimed
EP-4673584-A1 SOLID MOLDED SULFITE-BASED OXYGEN SCAVENGER COMPOSITION AND METHOD OF MANUFACTURE NCH Corporation (US) 2026-01-07 EP disclosed
WO-2024182716-A1 SOLID MOLDED SULFITE-BASED OXYGEN SCAVENGER COMPOSITION AND METHOD OF MANUFACTURE NCH CORPORATION (US) 2024-09-06 WO disclosed
US-20240295031-A1 Solid Molded Sulfite-Based Oxygen Scavenger Composition and Method of Manufacutre THE BANK OF NEW YORK MELLON TRUST COMPANY, N.A., AS NOTES COLLATERAL AGENT 2024-09-05 US disclosed
EP-4262824-A1 MULTICOMPONENT COMPOSITION COMPRISING SUCROSE SULFATE, ALGINATE, GELLAN GUM FOR THE TREATMENT OF GASTRIC REFLUX Drugs Minerals and Generics Italia S.R.L. In Forma Abbreviata D.M.G. Italia S.R.L. (IT) 2023-10-25 EP disclosed
CN-116462679-A Pyrazolopyrimidine derivative and application thereof in medicine 四川海思科制药有限公司 2023-07-21 CN disclosed
WO-2022130359-A1 MULTICOMPONENT COMPOSITION COMPRISING SUCROSE SULFATE, ALGINATE, GELLAN GUM FOR THE TREATMENT OF GASTRIC REFLUX DRUGS MINERALS AND GENERICS ITALIA S.R.L. IN FORMA ABBREVIATA D.M.G. ITALIA S.R.L. (IT) 2022-06-23 WO disclosed
CN-106754428-B Poria cocos mycelium liquid fermentation method 华中农业大学 2020-02-21 CN disclosed
CN-109414442-A (S) liquid preparation of-N- (5- ((R) -2- (2,5- difluorophenyl)-pyrrolidin-1-yl)-pyrazolo [1,5-A] pyrimidin-3-yl) -3- hydroxyl pyrrolidine -1- formamide 洛克索肿瘤学股份有限公司 2019-03-01 CN disclosed
CN-109310694-A METHODS OF TREATING PEDIATRIC CANCERS 洛克索肿瘤学股份有限公司 2019-02-05 CN disclosed
EP-1806333-A1 A method for manufacturing dialkyl carbonate GENERAL ELECTRIC COMPANY (US) 2007-07-11 EP disclosed
EP-1299341-B1 A METHOD FOR MANUFACTURING DIALKYL CARBONATE GEN ELECTRIC (US) 2007-04-25 EP disclosed
EP-1299341-A2 A METHOD FOR MANUFACTURING DIALKYL CARBONATE GENERAL ELECTRIC COMPANY (US) 2003-04-09 EP disclosed
US-6458914-B2 REACTING CARBON MONOXIDE, OXYGEN AND ALCOHOL IN THE PRESENCE OF A CATALYST PRODUCED BY REACTING TOGETHER AND INCLUDING A CUPRIC HALIDE AND AN ALKOXIDE COMPOUND OF A GROUP III THROUGH VII METAL; EFFICIENCY; ANTIFOULING AGENTS GENERAL ELECTRIC COMPANY 2002-10-01 US disclosed
EP-1189870-A1 METHOD FOR MANUFACTURING DIALKYL CARBONATE GENERAL ELECTRIC COMPANY (US) 2002-03-27 EP disclosed
US-20020007087-A1 Method for manufacturing dialkyl carbonate SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2002-01-17 US disclosed
WO-2002000596-A2 A METHOD FOR MANUFACTURING DIALKYL CARBONATE GENERAL ELECTRIC COMPANY (US) 2002-01-03 WO disclosed
US-6258923-B1 REACTING CARBON MONOXIDE, OXYGEN AND ALCOHOL GENERAL ELECTRIC COMPANY 2001-07-10 US disclosed
WO-2000076950-A1 METHOD FOR MANUFACTURING DIALKYL CARBONATE GENERAL ELECTRIC COMPANY (US) 2000-12-21 WO disclosed