Troclosene

Troclosene

SCHEMBL3872688

O.O.O=c1[nH]c(=O)n(Cl)c(=O)n1Cl

nearest known ligand 0.30

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Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Troclosene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Troclosene SCHEMBL6894267 1.00 APEX1 (0.30) APEX1
Troclosene SCHEMBL28991821 0.97
Troclosene SCHEMBL31099328 0.97
Troclosene SCHEMBL166386 0.97 APEX1 (0.31) APEX1
Troclosene SCHEMBL21745 0.94 APEX1 (0.30) APEX1
Troclosene SCHEMBL305053 0.94 APEX1 (0.30) APEX1
Troclosene SCHEMBL30616181 0.94 APEX1 (0.30) APEX1
Troclosene SCHEMBL531397 0.94 APEX1 (0.30) APEX1
Troclosene SCHEMBL9083160 0.94 APEX1 (0.30) APEX1
Troclosene SCHEMBL29779771 0.94 APEX1 (0.30) APEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7465410-B2 Solvent-activated reactor TRUOX, INC. (US) 2008-12-16 US claimed
US-20060197056-A1 Water soluble mixture that generates chlorine dioxide including chlorite donor and a free halogen donor, forms gel when exposed to the main solvent that encloses the reactants, restricts reactant diffusion, and prevents contact with solvent; ClO2 released through colloidal gel wall at a controlled rate TRUOX, INC. 2006-09-07 US claimed
WO-2006020247-A2 A SOLVENT-ACTIVATED REACTOR TRUOX, INC. (US) 2006-02-23 WO claimed
US-20060013751-A1 Solvent-activated reactor TRUOX, INC. 2006-01-19 US claimed
US-20040135116-A1 Massive bodies containing free halogen source for producing highly converted solutions of chlorine dioxide ENGELHARD CORPORATION 2004-07-15 US claimed
US-6699404-B2 TABLET, FOR PRODUCING A SOLUTION OF CHLORINE DIOXIDE WHEN THE MASSIVE BODY IS ADDED TO LIQUID WATER ENGELHARD CORPORATION 2004-03-02 US claimed
US-20030080317-A1 Massive bodies containing free halogen source for producing highly converted solutions of chlorine dioxide ENGELHARD CORPORATION 2003-05-01 US claimed
WO-2013036601-A1 USE OF MOSS TO REDUCE DISINFECTION BY-PRODUCTS IN WATER TREATED WITH DISINFECTANTS EMBRO CORPORATION (US) 2013-03-14 WO disclosed
CN-101448863-A Polyvinyl alcohol films with improved resistance to oxidizing chemicals CELANESE INT CORP (US) 2009-06-03 CN disclosed
US-7534368-B2 Water soluble mixture that generates chlorine dioxide including chlorite donor and a free halogen donor, forms gel when exposed to the main solvent that encloses the reactants, restricts reactant diffusion, and prevents contact with solvent; ClO2 released through colloidal gel wall at a controlled rate TRUOX, INC. (US) 2009-05-19 US disclosed
US-7514019-B2 Water soluble mixture that generates chlorine dioxide including chlorite donor and polymeric that forms a gel when exposed to the main solvent that encloses the reactants, restricts reactant diffusion, and prevents contact with solvent; ClO2 released through colloidal gel wall at a controlled rate TRUOX, INC. (US) 2009-04-07 US disclosed
US-7465410-B2 Solvent-activated reactor TRUOX, INC. (US) 2008-12-16 US disclosed
US-20060197056-A1 Water soluble mixture that generates chlorine dioxide including chlorite donor and a free halogen donor, forms gel when exposed to the main solvent that encloses the reactants, restricts reactant diffusion, and prevents contact with solvent; ClO2 released through colloidal gel wall at a controlled rate TRUOX, INC. 2006-09-07 US disclosed
US-20060013751-A1 Solvent-activated reactor TRUOX, INC. 2006-01-19 US disclosed
US-20060014872-A1 Protective composition that allows in-situ generation of permeation channels therein TRUOX, INC. 2006-01-19 US disclosed
US-20050155936-A1 Halogen-enhanced oxidizing composition TRUOX, INC. 2005-07-21 US disclosed
EP-0291097-B1 METHOD OF PREPARING SPHERICAL GRANULES AND TABLETS OF A SOLID CHLORINATING AGENT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1991-12-04 EP disclosed
EP-0291097-A2 Method of preparing spherical granules and tablets of a solid chlorinating agent NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1988-11-17 EP disclosed
US-4329431-A Instant culture media and method of sterilizing same YOUSSEF KAMAL A 1982-05-11 US disclosed
US-4248971-A ADDING CHLORINE-LIBERATING COMPOUND, WITHOUT AUTOCLAVING YOUSSEF KAMAL A 1981-02-03 US disclosed