SCHEMBL3884130

SCHEMBL3884130

C[C@H](NS(=O)(=O)c1ccc(Cl)cc1)C(=O)Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 7/20 0.57
MMP1 P03956 4/20 0.57
MMP9 P14780 4/20 0.57
MMP13 P45452 4/20 0.57
MMP3 P08254 3/20 0.57
MMP7 P09237 3/20 0.57
CA2 P00918 5/20 0.54
CA12 O43570 3/20 0.54
CA9 Q16790 3/20 0.54
CA14 Q9ULX7 3/20 0.54
SLC1A3 P43003 1/20 0.53
SLC1A2 P43004 1/20 0.53
SLC1A1 P43005 1/20 0.53
MMP8 P22894 3/20 0.52
MMP14 P50281 1/20 0.52
CA1 P00915 4/20 0.52
CA3 P07451 1/20 0.52
CA4 P22748 1/20 0.52
CA6 P23280 1/20 0.52
CA5A P35218 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3884127 1.00 MMP2 (0.57) MMP2MMP1MMP9MMP13MMP3
SCHEMBL5734780 0.86 TSHR (0.56) MMP2MMP1MMP9MMP13MMP3
SCHEMBL3951678 0.86 ADAMTS4 (0.69) MMP2MMP1MMP9MMP13MMP3
SCHEMBL5734792 0.86 TSHR (0.56) MMP2MMP1MMP9MMP13MMP3
SCHEMBL13890464 0.86 MMP2 (0.57) MMP2MMP1MMP9MMP13MMP3
SCHEMBL4380323 0.86 ADAMTS4 (0.69) MMP2MMP1MMP9MMP13MMP3
SCHEMBL28502922 0.86 TSHR (0.56) MMP2MMP1MMP9MMP13MMP3
SCHEMBL3951681 0.86 ADAMTS4 (0.69) MMP2MMP1MMP9MMP13MMP3
SCHEMBL6325782 0.84 ADAMTS4 (0.61) MMP2MMP1MMP9MMP13MMP3
SCHEMBL2337573 0.83 ALDH1A1 (0.56) MMP2MMP1MMP9MMP13MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090111860-A1 SULFONAMIDE COMPOUNDS USEFUL AS ADG RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2009-04-30 US disclosed
EP-2013184-A1 SULFONAMIDE COMPOUNDS USEFUL AS EDG RECEPTOR MODULATORS AstraZeneca AB (SE) 2009-01-14 EP disclosed
WO-2007129019-A1 SULFONAMIDE COMPOUNDS USEFUL AS EDG RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-11-15 WO disclosed
EP-1378507-B1 Process for producing optically active imidazole derivatives, intermediates and synthesis thereof MITSUBISHI PHARMA CORP (JP) 2006-08-23 EP disclosed
EP-1378507-A2 Process for producing optically active imidazole compounds, intermediates for synthesizing the same, and process for producing the same Mitsubishi Pharma Corporation (JP) 2004-01-07 EP disclosed
CN-1133623-C Process for producing optically active imidazole compound, intermediate for synthesis thereof, and process for producing the same ������ҩ��ʽ���� 2004-01-07 CN disclosed
US-6166221-A Production method of optically active imidazole compound, synthetic intermediate therefor and production method thereof YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
US-6066739-A Process for producing optically active imidazole compounds, intermediates for synthesizing the same, and process for producing the same YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2000-05-23 US disclosed
CN-1251093-A Process for producing optically active imidazole compound, intermediates for synthesizing same YOSHITOMI PHARMACEUTICAL (JP) 2000-04-19 CN disclosed
EP-0972768-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE IMIDAZOLE COMPOUNDS, INTERMEDIATES FOR SYNTHESIZING THE SAME, AND PROCESS FOR PRODUCING THE SAME YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2000-01-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090111860-A1 SULFONAMIDE COMPOUNDS USEFUL AS ADG RECEPTOR MODULATORS ADGRE5, ADGRF1, SELPLG MMP2 3625/4885MMP1 2733/4885MMP9 3153/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.