SCHEMBL3935197

SCHEMBL3935197

CCCCCc1cc(C)nn2c(-c3sc(Br)cc3OC)c(C)nc12

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 9/20 0.35
PI4KB Q9UBF8 1/20 0.35
CRHR1 P34998 5/20 0.34
CRHR2 Q13324 1/20 0.33
ALOX5 P09917 4/20 0.32
PTGS2 P35354 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3921099 0.79 CRHR1 (0.55) SMPD3PI4KBCRHR1CRHR2
SCHEMBL4787114 0.77 TLR8 (0.38) SMPD3CRHR1CRHR2
SCHEMBL4689862 0.76 CRHR1 (0.45) SMPD3CRHR1
SCHEMBL4690582 0.71 CRHR1 (0.53) CRHR1CRHR2
SCHEMBL4693477 0.71 CRHR1 (0.67) CRHR1CRHR2
SCHEMBL4693619 0.71 CRHR1 (0.67) CRHR1CRHR2
SCHEMBL4694319 0.70 CRHR1 (0.37) CRHR1CRHR2
SCHEMBL4694546 0.70 CRHR1 (0.39) CRHR1CRHR2
SCHEMBL4695462 0.69 ADRA2A (0.43) CRHR1ALOX5
SCHEMBL3920616 0.69 CRHR1 (0.57) SMPD3PI4KBCRHR1CRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869049-B1 IMIDAZOPYRIDAZINE COMPOUNDS LILLY CO ELI (US) 2009-03-04 EP disclosed