SCHEMBL3936397

SCHEMBL3936397

COC(=O)Cc1cccc(C2CCCN(S(=O)(=O)CCc3ccccc3)C2)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.45
DRD3 P35462 4/20 0.45
DRD1 P21728 2/20 0.45
DRD4 P21917 2/20 0.45
DRD5 P21918 2/20 0.45
MMP8 P22894 2/20 0.44
MMP12 P39900 2/20 0.44
MMP13 P45452 2/20 0.44
MMP1 P03956 1/20 0.44
MMP7 P09237 1/20 0.44
FKBP1A P62942 4/20 0.43
BCL9 O00512 2/20 0.43
CTNNB1 P35222 2/20 0.43
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3930618 0.90 ALDH1A1 (0.53) BCL9CTNNB1ALDH1A1HSD17B10HTT
SCHEMBL3930804 0.89 DRD2 (0.46) DRD2DRD3DRD1DRD4DRD5
SCHEMBL3939609 0.89 DRD3 (0.45) DRD2DRD3DRD1DRD4DRD5
SCHEMBL3943769 0.86 DRD2 (0.45) DRD2DRD3DRD1DRD4DRD5
Ethylbenzene SCHEMBL27747313 0.84 ALDH1A1 (0.40) DRD2DRD3DRD1DRD4DRD5
Chlorobenzene SCHEMBL27747004 0.83 BCL9 (0.39) DRD2DRD3DRD1DRD4DRD5
Anisole SCHEMBL27747003 0.83 ALDH1A1 (0.43) DRD2DRD3DRD1DRD4DRD5
Fluorobenzene SCHEMBL27747012 0.83 DRD2 (0.39) DRD2DRD3DRD1DRD4DRD5
1,2-Dichlorobenzene SCHEMBL27747023 0.82 ALDH1A1 (0.38) DRD2DRD3DRD1DRD4DRD5
SCHEMBL3935500 0.82 BCL9 (0.46) DRD2DRD3BCL9CTNNB1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044017-A2 SUBSTITUTED PHENYL ACETIC ACIDS AS DP-2 ANTAGONISTS ICOS CORPORATION (US) 2009-04-08 EP disclosed
WO-2007146838-A2 SUBSTITUTED PHENYL ACETIC ACIDS AS DP-2 ANTAGONISTS ICOS CORPORATION (US) 2007-12-21 WO disclosed