SCHEMBL3930618

SCHEMBL3930618

COC(=O)Cc1cccc(C2CCCN(S(=O)(=O)Cc3ccccc3)C2)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.53
HSD17B10 Q99714 2/20 0.53
MAPT P10636 4/20 0.50
NPSR1 Q6W5P4 3/20 0.50
HPGD P15428 2/20 0.50
LMNA P02545 3/20 0.46
MEN1 O00255 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
BCL9 O00512 1/20 0.44
CTNNB1 P35222 1/20 0.44
TSHR P16473 2/20 0.44
PKM P14618 2/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3936397 0.90 DRD2 (0.45) ALDH1A1HSD17B10HTTSMN1; SMN2BCL9
SCHEMBL3933032 0.89 ALDH1A1 (0.54) ALDH1A1HSD17B10MAPTNPSR1HPGD
SCHEMBL3943769 0.88 DRD2 (0.45) ALDH1A1MEN1KMT2ABCL9CTNNB1
SCHEMBL3939609 0.86 DRD3 (0.45) ALDH1A1HTTSMN1; SMN2TSHRPOLB
Ethylbenzene SCHEMBL27747313 0.85 ALDH1A1 (0.40) ALDH1A1HSD17B10MAPTMEN1KMT2A
Fluorobenzene SCHEMBL27747012 0.85 DRD2 (0.39) ALDH1A1HSD17B10NPSR1LMNABCL9
Anisole SCHEMBL27747003 0.85 ALDH1A1 (0.43) ALDH1A1HSD17B10HPGDLMNASMN1; SMN2
Chlorobenzene SCHEMBL27747004 0.85 BCL9 (0.39) ALDH1A1HSD17B10BCL9CTNNB1
1,2-Dichlorobenzene SCHEMBL27747023 0.84 ALDH1A1 (0.38) ALDH1A1HSD17B10MAPTNPSR1HPGD
SCHEMBL3935500 0.83 BCL9 (0.46) MAPTLMNAMEN1KMT2ABCL9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044017-A2 SUBSTITUTED PHENYL ACETIC ACIDS AS DP-2 ANTAGONISTS ICOS CORPORATION (US) 2009-04-08 EP disclosed
WO-2007146838-A2 SUBSTITUTED PHENYL ACETIC ACIDS AS DP-2 ANTAGONISTS ICOS CORPORATION (US) 2007-12-21 WO disclosed