SCHEMBL3942136

SCHEMBL3942136

Nc1ccc2[nH]c(OC(=O)Nc3ccccn3)c(-c3ccccc3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
PKM P14618 2/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A3 Q01959 1/20 0.37
FLT3 P36888 2/20 0.37
STK17B O94768 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
GSK3B P49841 1/20 0.37
ADK P55263 1/20 0.37
PADI4 Q9UM07 2/20 0.37
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3947601 0.85 BRD4 (0.42) MEN1KMT2AFLT3STK17BCDK5
SCHEMBL3945191 0.84 MAPT (0.53) NPC1RAB9AMEN1KMT2APKM
SCHEMBL4924331 0.82 ALDH1A1 (0.51) NPC1RAB9AMEN1KMT2ACHRNB2
SCHEMBL5187596 0.82 NPC1 (0.41) NPC1RAB9APKMPADI4ALDH1A1
SCHEMBL3943641 0.78 LHCGR (0.44) RAB9AGSK3BADKALDH1A1KDM4E
SCHEMBL3951863 0.77 ALDH1A1 (0.43) MEN1KMT2AFLT3STK17BCDK5
SCHEMBL3946458 0.76 BRD4 (0.49) MEN1KMT2AALDH1A1KDM4E
SCHEMBL3951513 0.74 HTR2C (0.39) MEN1KMT2AGSK3BADKPADI4
SCHEMBL3946744 0.73 LIPE (0.41) MEN1KMT2AGSK3BADKALDH1A1
SCHEMBL3943442 0.70 ALDH1A1 (0.47) KMT2APADI4ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802572-B1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE BAYER SCHERING PHARMA AG (DE) 2009-04-22 EP disclosed
EP-1802572-A1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE Bayer Schering Pharma Aktiengesellschaft (DE) 2007-07-04 EP disclosed
WO-2006032541-A1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-03-30 WO disclosed