SCHEMBL3947601

SCHEMBL3947601

Nc1ccc2[nH]c(OC(=O)Nc3ccccc3)c(-c3ccccc3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.42
GSK3B P49841 2/20 0.41
ADK P55263 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 3/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
MAP2 P11137 3/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NGFR P08138 1/20 0.39
FLT3 P36888 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
STK17B O94768 1/20 0.38
CDK5 Q00535 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5187596 0.90 NPC1 (0.41) ALDH1A1KDM4EGAAMAPTDYRK1A
SCHEMBL3942136 0.85 NPC1 (0.39) GSK3BADKALDH1A1KDM4EGAA
SCHEMBL3943641 0.83 LHCGR (0.44) GSK3BADKALDH1A1KDM4EGAA
SCHEMBL3951863 0.82 ALDH1A1 (0.43) GSK3BADKALDH1A1KDM4EGAA
SCHEMBL3948652 0.82 MAPT (0.60) GSK3BALDH1A1KDM4EMAPTKMT2A
SCHEMBL3951020 0.80 FAAH (0.50) ALDH1A1
SCHEMBL3951513 0.79 HTR2C (0.39) GSK3BADKALDH1A1KDM4EGAA
SCHEMBL4929236 0.79 ALDH1A1 (0.57) ALDH1A1KDM4EGAAMAPTMAP2
SCHEMBL3946744 0.79 LIPE (0.41) GSK3BADKALDH1A1KDM4EGAA
SCHEMBL3942565 0.76 PTGS2 (0.44) BRD4KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802572-B1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE BAYER SCHERING PHARMA AG (DE) 2009-04-22 EP disclosed
EP-1802572-A1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE Bayer Schering Pharma Aktiengesellschaft (DE) 2007-07-04 EP disclosed
WO-2006032541-A1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-03-30 WO disclosed