SCHEMBL3955545

SCHEMBL3955545

c1ccc(CNc2cnccn2)nc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.65
HPGD P15428 5/20 0.65
MEN1 O00255 2/20 0.65
KMT2A Q03164 2/20 0.65
MAOA P21397 3/20 0.56
MAOB P27338 3/20 0.56
KDM4E B2RXH2 6/20 0.54
NPC1 O15118 3/20 0.54
RAB9A P51151 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TP53 P04637 1/20 0.54
HTT P42858 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
CXCR4 P61073 1/20 0.49
FYN P06241 1/20 0.48
FABP1 P07148 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL229311 0.83 CXCR4 (0.68) ALDH1A1HPGDMEN1KMT2AMAOA
SCHEMBL30487250 0.83 CXCR4 (0.68) ALDH1A1HPGDMEN1KMT2AMAOA
SCHEMBL3953451 0.79 ALDH1A1 (1.00) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL1239720 0.79 CHRM2 (0.56) ALDH1A1MEN1KMT2AMAOAMAOB
SCHEMBL18949331 0.77 ALDH1A1 (0.53) ALDH1A1HPGDMEN1KMT2AMAOA
SCHEMBL1244338 0.75 MAOA (0.70) ALDH1A1HPGDMEN1KMT2AMAOA
SCHEMBL12198925 0.75 MAOA (0.54) ALDH1A1HPGDMEN1KMT2AMAOA
SCHEMBL3948160 0.74 ALDH1A1 (0.77) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL29846220 0.74 MAOA (0.68) ALDH1A1HPGDMEN1KMT2AMAOA
SCHEMBL23938004 0.73 NPC1 (0.62) ALDH1A1HPGDMEN1KMT2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029617-A1 DIARYLAMINE-SUBSTITUTED QUINOLONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed