SCHEMBL3963960

SCHEMBL3963960

Cc1nc2ccc(N3CCCCC3)cc2c(-c2ccc(F)cc2)c1CCOc1ccccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.42
SLC2A1 P11166 1/20 0.40
KCNH2 Q12809 1/20 0.40
HTT P42858 1/20 0.39
TSHR P16473 1/20 0.38
ELOVL1 Q9BW60 1/20 0.38
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
IDO2 Q6ZQW0 1/20 0.37
KDM4E B2RXH2 3/20 0.37
METTL3 Q86U44 1/20 0.37
METTL14 Q9HCE5 1/20 0.37
MAPT P10636 4/20 0.36
RAB9A P51151 1/20 0.36
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
LMNA P02545 1/20 0.36
SMO Q99835 1/20 0.36
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3970453 0.88 L3MBTL1 (0.38) ELOVL1IDO1TDO2IDO2KDM4E
SCHEMBL3958654 0.87 MAPT (0.36) HTTELOVL1IDO1TDO2IDO2
SCHEMBL3963734 0.87 DRD2 (0.45) MCHR1KCNH2ELOVL1IDO1TDO2
SCHEMBL3970359 0.86 ELOVL1 (0.46) KCNH2ELOVL1IDO1TDO2IDO2
SCHEMBL4198373 0.84 KCNH2 (0.39) MCHR1KCNH2ELOVL1
SCHEMBL3969490 0.84 KCNH2 (0.41) KCNH2KDM4EMAPTLMNASMO
SCHEMBL3964828 0.83 KCNH2 (0.43) KCNH2TSHRELOVL1IDO1TDO2
SCHEMBL3962203 0.83 ELOVL1 (0.39) KCNH2ELOVL1IDO1TDO2IDO2
SCHEMBL3962968 0.82 IDO1 (0.42) ELOVL1IDO1TDO2IDO2KDM4E
SCHEMBL3966727 0.82 PIK3CD (0.40) KCNH2TSHRELOVL1IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041904-A1 QUINOLINE COMPOUNDS HAVING AN ACTIVITY AGAINST THE GABAB RECEPTOR ASTRAZENECA AB (SE) 2009-04-02 WO claimed
WO-2009041904-A1 QUINOLINE COMPOUNDS HAVING AN ACTIVITY AGAINST THE GABAB RECEPTOR ASTRAZENECA AB (SE) 2009-04-02 WO disclosed