SCHEMBL3968052

SCHEMBL3968052

Cc1c(Cl)cc2c(c1-c1ccccc1)C(=O)[C@H](N1CCNCC1)C(=O)N2Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.36
SIGMAR1 Q99720 1/20 0.35
ALDH1A1 P00352 8/20 0.35
TACR1 P25103 1/20 0.35
MAPK1 P28482 2/20 0.34
USP2 O75604 4/20 0.34
GAA P10253 3/20 0.34
TP53 P04637 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
EGFR P00533 1/20 0.33
POLB P06746 2/20 0.33
ALOX15 P16050 2/20 0.33
CHRM3 P20309 1/20 0.33
MAPT P10636 2/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8231306 0.69 CES2 (0.42) HTR6ALDH1A1TP53MEN1KMT2A
SCHEMBL8910312 0.67 DRD4 (0.41) ALDH1A1MEN1KMT2ACHRM3MAPT
SCHEMBL8910768 0.67 DRD4 (0.39) ALDH1A1MEN1KMT2AMAPTDRD2
SCHEMBL4674919 0.60 HTR6 (0.64) HTR6SIGMAR1ALDH1A1MEN1KMT2A
SCHEMBL4675159 0.60 HTR6 (0.64) HTR6SIGMAR1ALDH1A1MEN1KMT2A
SCHEMBL4675195 0.60 HTR6 (0.64) HTR6SIGMAR1ALDH1A1MEN1KMT2A
Aziridine SCHEMBL29206308 0.59 SIGMAR1 (0.50) HTR6SIGMAR1ALDH1A1GAAMEN1
SCHEMBL6781872 0.59 KMT2A (0.58) ALDH1A1MAPK1USP2GAAMEN1
SCHEMBL584720 0.57 ALDH1A1 (0.69) ALDH1A1MAPK1MEN1KMT2A
SCHEMBL5770320 0.57 ALDH1A1 (0.69) ALDH1A1MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954689-A4 N-SUBSTITUTED-1H-QUINOLINE-2, 4-DIONES, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RES INST CHEM TECH (KR) 2009-09-02 EP disclosed
EP-1954689-A1 N-SUBSTITUTED-1H-QUINOLINE-2, 4-DIONES, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2008-08-13 EP disclosed
WO-2007032572-A1 N-SUBSTITUTED-1H-QUINOLINE-2, 4-DIONES, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KOREA RESERACH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2007-03-22 WO disclosed