SCHEMBL3971153

SCHEMBL3971153

CCOc1cc(CN(c2ccc(C#N)cc2)C2CCNCC2)ccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 11/20 0.52
SLC6A2 P23975 10/20 0.52
SLC6A3 Q01959 8/20 0.52
NOS2 P35228 4/20 0.44
CYP19A1 P11511 1/20 0.39
NOS3 P29474 3/20 0.39
NOS1 P29475 3/20 0.39
CCR5 P51681 1/20 0.39
HTR6 P50406 1/20 0.37
TACR1 P25103 1/20 0.37
PGR P06401 1/20 0.37
S1PR1 P21453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973450 0.88 SLC6A2 (0.52) SLC6A4SLC6A2SLC6A3NOS2CYP19A1
SCHEMBL3976469 0.86 SLC6A2 (0.40) SLC6A4SLC6A2SLC6A3NOS2NOS3
SCHEMBL3973780 0.84 SLC6A2 (0.40) SLC6A4SLC6A2SLC6A3NOS2NOS3
SCHEMBL3971824 0.80 NOS2 (0.41) SLC6A4SLC6A2SLC6A3NOS2NOS3
SCHEMBL4701500 0.79 SLC6A2 (0.41) SLC6A4SLC6A2SLC6A3NOS2NOS3
SCHEMBL5558707 0.78 SLC6A2 (0.48) SLC6A4SLC6A2SLC6A3HTR6TACR1
SCHEMBL3997957 0.78 TACR1 (0.39) SLC6A4SLC6A2SLC6A3TACR1
SCHEMBL4544203 0.77 SLC6A2 (0.45) SLC6A4SLC6A2SLC6A3
SCHEMBL3977938 0.76 RORC (0.44) SLC6A4SLC6A2SLC6A3TACR1S1PR1
SCHEMBL3973733 0.76 SLC6A2 (0.39) SLC6A4SLC6A2SLC6A3NOS2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed