SCHEMBL3976494

SCHEMBL3976494

CC(C)c1ccc(C(=O)NCCCCc2cn(-c3ccccc3)c3ccc(C(=O)O)cc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
LMNA P02545 1/20 0.44
HDAC3 O15379 1/20 0.44
HPGD P15428 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
PTAFR P25105 3/20 0.42
PLA2G4A P47712 4/20 0.42
MAPK8 P45983 2/20 0.42
SCN2B O60939 1/20 0.40
SCN1A P35498 1/20 0.40
SCN1B Q07699 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
RORC P51449 1/20 0.40
TBXAS1 P24557 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3971346 0.92 NPC1 (0.44) NPC1RAB9ASMN1; SMN2LMNAHPGD
SCHEMBL13883740 0.89 NPC1 (0.48) NPC1RAB9ASMN1; SMN2MTNR1AMTNR1B
SCHEMBL3971172 0.88 PTAFR (0.48) NPC1RAB9ASMN1; SMN2LMNAHDAC3
SCHEMBL3971256 0.88 NPC1 (0.47) NPC1RAB9ASMN1; SMN2MTNR1AMTNR1B
SCHEMBL13883686 0.87 RORC (0.45) NPC1RAB9ASMN1; SMN2MTNR1AMTNR1B
SCHEMBL3972294 0.87 NAMPT (0.48) MTNR1AMTNR1BHDAC3HDAC1HDAC2
SCHEMBL13883906 0.84 TMEM97 (0.45) NPC1RAB9ASMN1; SMN2MTNR1AMTNR1B
SCHEMBL3975570 0.84 RAB9A (0.47) RAB9AMTNR1AMTNR1BLMNAHDAC3
SCHEMBL3970351 0.83 MTNR1A (0.51) MTNR1AMTNR1BHPGDPLA2G4A
SCHEMBL13883750 0.83 ABCB1 (0.42) NPC1RAB9ASMN1; SMN2LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO claimed
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed