SCHEMBL3973590

SCHEMBL3973590

Oc1cccc(-n2nnc(S)c2-c2ccccc2-c2ccccc2)c1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNMA1 Q12791 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
BCL2L1 Q07817 1/20 0.38
HSD17B10 Q99714 1/20 0.38
BRD4 O60885 1/20 0.37
NR1I2 O75469 1/20 0.37
SMARCA2 P51531 1/20 0.37
SMARCA4 P51532 1/20 0.37
PBRM1 Q86U86 1/20 0.37
DHODH Q02127 3/20 0.36
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
KCNN4 O15554 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
GAA P10253 1/20 0.33
GFER P55789 1/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1148629 0.81 ALOX5 (0.44) KCNMA1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL4088457 0.79 KCNMA1 (0.36) KCNMA1BRD4MAPTKDM4EPOLB
SCHEMBL4077177 0.78 KDM4E (0.39) KCNMA1ALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL3974239 0.77 KCNMA1 (0.36) KCNMA1CCNE1CDK2RAB9AMEN1
SCHEMBL3974759 0.77 MAPK9 (0.41) KCNMA1CCNE1CDK2MAPK10
SCHEMBL3973703 0.76 KCNN4 (0.37) KCNMA1ALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL4089989 0.76 MGAM (0.35) KCNMA1KCNN4GAA
SCHEMBL5329381 0.76 TRPA1 (0.40) KCNMA1ALDH1A1GAA
SCHEMBL3974423 0.75 KDM4E (0.36) KCNMA1ALDH1A1CDK2KDM4EKMT2A
SCHEMBL1148311 0.75 KCNMA1 (0.46) KCNMA1ALDH1A1HPGDHSD17B10DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054059-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-05-06 EP claimed
WO-2008021364-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-02-21 WO claimed