SCHEMBL3974239

SCHEMBL3974239

Oc1cccc(-n2nnc(S)c2-c2ccc(Cl)cc2)c1O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNMA1 Q12791 1/20 0.36
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA4 P22748 4/20 0.34
CA9 Q16790 4/20 0.34
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
PDE4B Q07343 1/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3974759 0.81 MAPK9 (0.41) KCNMA1CA1CA2CA9CCNE1
SCHEMBL1148724 0.78 MEN1 (0.37) CA1CA2CA4CA9MEN1
SCHEMBL3973590 0.77 KCNMA1 (0.38) KCNMA1MEN1RAB9AKMT2ACCNE1
SCHEMBL4088457 0.77 KCNMA1 (0.36) KCNMA1
SCHEMBL5329381 0.77 TRPA1 (0.40) KCNMA1TP53
SCHEMBL1148519 0.75 KCNMA1 (0.48) KCNMA1CA1CA2CA4CA9
SCHEMBL1148472 0.75 KCNMA1 (0.48) KCNMA1CA1CA2CA4CA9
SCHEMBL5369428 0.74 GABRA1 (0.37) KCNMA1CA1CA2TP53
SCHEMBL3974423 0.71 KDM4E (0.36) KCNMA1KMT2ACDK2
SCHEMBL1148326 0.70 ALOX5 (0.37) CA9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054059-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-05-06 EP claimed
WO-2008021364-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-02-21 WO claimed