SCHEMBL4089989

SCHEMBL4089989

Cc1[nH]c2cccc(-c3c(S)nnn3-c3cccc(O)c3O)c2c1C

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MGAM O43451 2/20 0.35
GAA P10253 2/20 0.35
SI P14410 2/20 0.35
MGAM2 Q2M2H8 2/20 0.35
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
KCNMA1 Q12791 1/20 0.32
F7 P08709 1/20 0.31
BTK Q06187 1/20 0.31
KCNN4 O15554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1148407 0.84 GAA (0.36) MGAMGAASIMGAM2BTK
SCHEMBL3973590 0.76 KCNMA1 (0.38) GAAKCNMA1KCNN4
SCHEMBL5329381 0.75 TRPA1 (0.40) MGAMGAASIMGAM2KCNMA1
SCHEMBL3973703 0.73 KCNN4 (0.37) GAAKCNMA1KCNN4
SCHEMBL3974423 0.72 KDM4E (0.36) KCNMA1
SCHEMBL4088457 0.71 KCNMA1 (0.36) KCNMA1
SCHEMBL5369428 0.70 GABRA1 (0.37) HTR2CKCNMA1
SCHEMBL3974239 0.69 KCNMA1 (0.36) KCNMA1
SCHEMBL3972617 0.69 NPC1 (0.38) GAA
SCHEMBL4077177 0.68 KDM4E (0.39) GAAKCNMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054059-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-05-06 EP claimed
WO-2008021364-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-02-21 WO claimed