SCHEMBL3973663

SCHEMBL3973663

C=C(O)CNC(=O)c1ccccc1C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
APEX1 P27695 1/20 0.45
TSHR P16473 2/20 0.42
HTT P42858 2/20 0.42
BCAT2 O15382 1/20 0.42
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KEAP1 Q14145 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2129167 0.82 TSHR (0.47) KMT2AAPEX1TSHRHTTBCAT2
SCHEMBL14839314 0.81 HPGD (0.55) KMT2ATSHRHTTKDM4EHPGD
SCHEMBL6903284 0.80 TSHR (0.58) KMT2AAPEX1TSHRHTTKDM4E
SCHEMBL9329299 0.77 TSHR (0.46) KMT2AAPEX1TSHRHTTBCAT2
SCHEMBL6566957 0.77 TSHR (0.55) KMT2AAPEX1TSHRHTTKDM4E
SCHEMBL6075765 0.77 TSHR (0.46) KMT2AAPEX1TSHRHTTBCAT2
SCHEMBL461826 0.76 HPGD (0.66) KMT2AKDM4EHPGDALDH1A1MAPT
SCHEMBL7870127 0.76 HPGD (0.66) KMT2AKDM4EHPGDALDH1A1MAPT
SCHEMBL1628440 0.76 GAA (0.63) HPGDALDH1A1MAPTHSD17B10NPC1
SCHEMBL31448014 0.75 KEAP1 (0.62) KMT2AAPEX1TSHRHTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1923436-B1 Powder compositions comprising Beta-Hydroxyalkyl amides from the ring-opening of acidic coumpounds ROHM & HAAS (US) 2009-01-21 EP disclosed
EP-1923436-A1 Powder compositions comprising Beta-Hydroxyalkyl amides from the ring-opening of acidic coumpounds Rohm and Haas Company (US) 2008-05-21 EP disclosed
US-20080114132-A1 Powder compositions comprising beta-hydroxyalkyl amides from the ring-opening of acidic compounds AKZO NOBEL COATINGS INTERNATIONAL B.V. (NL) 2008-05-15 US disclosed