SCHEMBL3973960

SCHEMBL3973960

Cc1cccc2c(C(=O)c3cc(Cl)ncn3)n(C)nc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
GLA P06280 1/20 0.38
SSTR4 P31391 1/20 0.35
BCL2 P10415 1/20 0.34
MCL1 Q07820 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CASP1 P29466 6/20 0.33
CASP7 P55210 6/20 0.33
HSD17B10 Q99714 5/20 0.33
MAPT P10636 3/20 0.33
HTT P42858 1/20 0.33
ALDH1A1 P00352 4/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
LCK P06239 1/20 0.32
HPGD P15428 3/20 0.32
TSHR P16473 2/20 0.32
RAB9A P51151 1/20 0.32
SLC22A12 Q96S37 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3972580 0.84 DHODH (0.33) KDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL3990181 0.75 RORC (0.39) L3MBTL1MCL1MEN1KMT2A
SCHEMBL9388097 0.74 SSTR4 (0.43) KDM4EL3MBTL1SSTR4MCL1SMN1; SMN2
SCHEMBL3973747 0.72 KMT2A (0.44) KDM4EL3MBTL1GLABCL2MCL1
SCHEMBL3979300 0.72 CDK2 (0.36) SMN1; SMN2HSD17B10MAPTHTTALDH1A1
SCHEMBL3972624 0.70 POLB (0.55) SMN1; SMN2MAPTHTTALDH1A1MEN1
SCHEMBL28242027 0.68 KMO (0.40) MEN1KMT2ALMNAKMO
SCHEMBL2260028 0.68 NPSR1 (0.41) KDM4EL3MBTL1MAPTALDH1A1MEN1
SCHEMBL3975153 0.67 NPC1 (0.38) L3MBTL1BCL2MCL1SMN1; SMN2MAPT
SCHEMBL3994459 0.67 PCSK9 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed