SCHEMBL3980764

SCHEMBL3980764

Cc1[nH]c2ccccc2c1-c1nsc2cc(F)ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 2/20 0.46
IMPDH2 P12268 1/20 0.43
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
MAPT P10636 4/20 0.42
ALDH1A1 P00352 4/20 0.42
GAA P10253 4/20 0.42
LMNA P02545 3/20 0.42
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
EIF2AK2 P19525 2/20 0.42
ATP4A P20648 2/20 0.42
ATP4B P51164 2/20 0.42
KDM4E B2RXH2 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CCR6 P51684 1/20 0.40
HKDC1 Q2TB90 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2961511 0.88 HTR7 (0.43) CYP1A2CYP2C9IMPDH2MEN1KMT2A
SCHEMBL317502 0.77 MEN1 (0.42) CYP1A2CYP2C9IMPDH2MEN1KMT2A
SCHEMBL2959702 0.75 KIF11 (0.48) CYP1A2CYP2C9MEN1KMT2AKDM4E
SCHEMBL317690 0.72 SMN1; SMN2 (0.35) CYP1A2CYP2C9IMPDH2MEN1KMT2A
SCHEMBL27701196 0.70 IMPDH2 (0.65) CYP1A2CYP2C9IMPDH2MEN1KMT2A
SCHEMBL704586 0.70 IMPDH2 (0.55) CYP1A2CYP2C9IMPDH2MEN1KMT2A
SCHEMBL1121782 0.68 CCNB2 (0.44) MAPTALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL1757795 0.68 HTR2A (0.43) CYP1A2CYP2C9IMPDH2MAPTALDH1A1
SCHEMBL12561582 0.66 MAPT (0.55) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL27681973 0.65 PTGS2 (0.59) IMPDH2MEN1KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805171-A4 INDOLE ACETIC ACIDS EXHIBITING CRTH2 RECEPTOR ANTAGONISM AND USES THEREOF WYETH CORP (US) 2009-05-13 EP disclosed
EP-1805171-A2 INDOLE ACETIC ACIDS EXHIBITING CRTH2 RECEPTOR ANTAGONISM AND USES THEREOF Athersys, Inc. (US) 2007-07-11 EP disclosed
WO-2006034419-A2 INDOLE ACETIC ACIDS EXHIBITING CRTH2 RECEPTOR ANTAGONISM AND USES THEREOF ATHERSYS, INC. (US) 2006-03-30 WO disclosed