SCHEMBL3989377

SCHEMBL3989377

CC(C)C(NCC(=O)OCc1ccccc1)C(=O)NC(Cc1ccc(O)c(C(C)(C)C)c1)CS(C)(=O)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.39
CA5A P35218 1/20 0.39
CA1 P00915 1/20 0.38
CASP3 P42574 2/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ABCC3 O15438 1/20 0.37
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
NR3C1 P04150 1/20 0.37
RARG P13631 1/20 0.37
CNR1 P21554 1/20 0.37
OPRK1 P41145 1/20 0.37
NR1H2 P55055 1/20 0.37
PPARA Q07869 1/20 0.37
NR1H3 Q13133 1/20 0.37
NR1I3 Q14994 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3987635 0.90 CA2 (0.38) CA2CA5ACA1CASP3CYP1A2
SCHEMBL3987632 0.85 CTSD (0.41) CA2CA5ACA1CASP3CYP1A2
SCHEMBL3989379 0.82 ABCB1 (0.36) CA2CA5ACA1CASP3CYP1A2
SCHEMBL4657183 0.78 CTSL (0.47) CA2CA5ACA1CTSDPSMB11
SCHEMBL3993261 0.77 PSMB11 (0.34) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3993264 0.77 MAPT (0.36) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7788731 0.77 CA4 (0.41) CA2CA5ACA1CASP3CTSD
SCHEMBL4656413 0.76 SYK (0.51) CA2CA5ACA1CTSD
SCHEMBL13795951 0.76 REN (0.34) OPRK1BACE1
SCHEMBL3987520 0.75 CTSL (0.41) CASP3OPRK1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed