SCHEMBL4004985

SCHEMBL4004985

COc1cc(-c2cnc(N)c(-c3nc4cc(S(N)(=O)=O)ccc4[nH]3)n2)ccc1OCCN1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 9/20 0.47
PRKDC P78527 1/20 0.46
ATM Q13315 1/20 0.46
ADORA2A P29274 2/20 0.45
ADORA1 P30542 1/20 0.45
MAP3K11 Q16584 3/20 0.43
MCHR1 Q99705 6/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4009811 0.88 MCHR1 (0.49) ATRADORA2AADORA1MAP3K11MCHR1
SCHEMBL4006573 0.87 ATR (0.59) ATRPRKDCATM
SCHEMBL4008321 0.86 ATR (0.55) ATRADORA2AADORA1MAP3K11MCHR1
SCHEMBL4009857 0.86 MCHR1 (0.51) ATRADORA2AADORA1MAP3K11MCHR1
SCHEMBL3927916 0.85 ATR (0.48) ATRADORA2AADORA1MAP3K11MCHR1
SCHEMBL4012928 0.81 ATR (0.54) ATRADORA2AADORA1MAP3K11MCHR1
SCHEMBL4297778 0.80 ATR (0.58) ATRPRKDCATMADORA2AMAP3K11
SCHEMBL4008973 0.75 ADORA2A (0.47) ADORA2AADORA1MAP3K11MCHR1
SCHEMBL3928126 0.73 MCHR1 (0.47) ADORA2AADORA1MAP3K11MCHR1
SCHEMBL4011105 0.73 MCHR1 (0.52) ATRADORA2AADORA1MAP3K11MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO disclosed